SCHEMBL17399321

SCHEMBL17399321

CC(=O)c1c(C2CC3CC[C@H](C2)N3C(=O)CO)nc2c(-c3ccc(-c4ncc[nH]4)nc3)cnn2c1N

nearest known ligand 0.56

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
MTOR P42345 15/20 0.56
RPTOR Q8N122 4/20 0.56
MLST8 Q9BVC4 4/20 0.56
CHEK1 O14757 4/20 0.33
CCNA2 P20248 4/20 0.33
CDK2 P24941 4/20 0.33
CCNA1 P78396 4/20 0.33
BRAF P15056 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2170325 1.00 MTOR (0.56) MTORRPTORMLST8CHEK1CCNA2
SCHEMBL2170333 1.00 MTOR (0.56) MTORRPTORMLST8CHEK1CCNA2
SCHEMBL2147872 1.00 MTOR (0.56) MTORRPTORMLST8CHEK1CCNA2
SCHEMBL12461531 1.00 MTOR (0.56) MTORRPTORMLST8CHEK1CCNA2
SCHEMBL14246212 0.94 MTOR (0.54) MTORRPTORMLST8CHEK1CCNA2
SCHEMBL14298609 0.94 MTOR (0.54) MTORRPTORMLST8CHEK1CCNA2
SCHEMBL2148172 0.94 MTOR (0.54) MTORRPTORMLST8CHEK1CCNA2
SCHEMBL2147123 0.94 MTOR (0.54) MTORRPTORMLST8CHEK1CCNA2
SCHEMBL14298598 0.94 MTOR (0.54) MTORRPTORMLST8CHEK1CCNA2
SCHEMBL14245926 0.94 MTOR (0.54) MTORRPTORMLST8CHEK1CCNA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9227971-B2 Pyrazolo[1,5-a]pyrimidine compounds as mTOR inhibitors MERCK SHARP & DOHME CORP. (US) 2016-01-05 US disclosed