SCHEMBL17399665

SCHEMBL17399665

CC(C(=N)NC(=O)c1cn(C2COC2)cn1)(c1ccc(-c2cnc(N)nc2)cc1)C1CC1

nearest known ligand 0.39

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
ALOX5AP P20292 19/20 0.39
CYP2C9 P11712 1/20 0.38
GSK3B P49841 1/20 0.36
DYRK1A Q13627 1/20 0.36
CYP2D6 P10635 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17399661 0.83 ALOX5AP (0.37) ALOX5APCYP2C9CYP2D6
SCHEMBL15166464 0.75 ALOX5AP (0.47) ALOX5APCYP2C9CYP2D6
SCHEMBL15166465 0.75 ALOX5AP (0.37) ALOX5APCYP2C9CYP2D6
SCHEMBL12005308 0.73 ALOX5AP (0.46) ALOX5APCYP2C9CYP2D6
SCHEMBL18220924 0.73 ALOX5AP (0.42) ALOX5APCYP2C9CYP2D6
SCHEMBL15166476 0.72 ALOX5AP (0.55) ALOX5APCYP2C9CYP2D6
SCHEMBL15166463 0.71 ALOX5AP (0.46) ALOX5APCYP2C9CYP2D6
SCHEMBL15166490 0.70 ALOX5AP (0.40) ALOX5APCYP2C9CYP2D6
SCHEMBL15166467 0.67 ALOX5AP (0.47) ALOX5APCYP2C9GSK3BDYRK1ACYP2D6
SCHEMBL670103 0.67 ALOX5AP (0.65) ALOX5APCYP2C9CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2606045-B1 OXADIAZOLE INHIBITORS OF LEUKOTRIENE PRODUCTION BOEHRINGER INGELHEIM INT (DE) 2016-01-06 EP disclosed