SCHEMBL1740299

SCHEMBL1740299

CC(=O)Nc1ccc(-c2nc(SCc3cccc(CCC(=O)N4CCN(CC5CCN(CCCO)C(I)C5)CC4)n3)nc(N)c2C#N)cc1

nearest known ligand 0.66

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
ADORA1 P30542 12/20 0.66
ADORA2A P29274 2/20 0.66
ADORA3 P0DMS8 1/20 0.32
ADORA2B P29275 1/20 0.32
IKBKB O14920 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL415216 0.91 ADORA1 (0.73) ADORA1ADORA2AADORA3ADORA2BIKBKB
SCHEMBL414307 0.89 ADORA1 (0.75) ADORA1ADORA2AADORA3ADORA2BIKBKB
SCHEMBL10135692 0.87 ADORA1 (0.74) ADORA1ADORA2AADORA3ADORA2B
SCHEMBL412422 0.86 ADORA1 (0.74) ADORA1ADORA2AADORA3ADORA2BIKBKB
Fumaric Acid SCHEMBL411630 0.86 ADORA1 (0.70) ADORA1ADORA2AADORA3ADORA2BIKBKB
Maleic Acid SCHEMBL411628 0.86 ADORA1 (0.70) ADORA1ADORA2AADORA3ADORA2BIKBKB
SCHEMBL414200 0.85 ADORA1 (0.73) ADORA1ADORA2AADORA3ADORA2B
SCHEMBL417963 0.85 ADORA1 (0.72) ADORA1ADORA2AADORA3ADORA2BIKBKB
Hydrochloric Acid SCHEMBL414128 0.84 ADORA1 (0.72) ADORA1ADORA2AADORA3ADORA2B
SCHEMBL945688 0.83 ADORA1 (0.83) ADORA1ADORA2AADORA3ADORA2BIKBKB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2393552-A1 A NOVEL CYANOPYRIMIDINE DERIVATIVE Otsuka Pharmaceutical Co., Ltd. (JP) 2011-12-14 EP claimed
WO-2010090299-A1 A NOVEL CYANOPYRIMIDINE DERIVATIVE OTSUKA PHARMACEUTICAL CO., LTD. (JP) 2010-08-12 WO claimed