SCHEMBL17409116

SCHEMBL17409116

CCc1cc(OCc2ccccc2)no1

nearest known ligand 0.48

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
SMPD1 P17405 1/20 0.47
BRD4 O60885 1/20 0.44
NPC1 O15118 1/20 0.43
RAB9A P51151 1/20 0.43
GABRA5 P31644 1/20 0.42
NUDT1 P36639 1/20 0.42
PKM P14618 1/20 0.42
MEN1 O00255 1/20 0.41
KMT2A Q03164 1/20 0.41
HCAR2 Q8TDS4 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15684128 0.83 SMPD1 (0.47) SMPD1BRD4NPC1RAB9AGABRA5
SCHEMBL25025302 0.83 SMPD1 (0.47) SMPD1BRD4NPC1RAB9AGABRA5
SCHEMBL322866 0.83 SMPD1 (0.53) SMPD1BRD4NPC1RAB9A
SCHEMBL12268217 0.83 SMPD1 (0.47) SMPD1BRD4NPC1RAB9AGABRA5
SCHEMBL13520120 0.83 NOTUM (0.51) SMPD1BRD4NPC1RAB9ANUDT1
SCHEMBL979239 0.83 SMPD1 (0.44) SMPD1BRD4
SCHEMBL28080632 0.81 SMPD1 (0.43) SMPD1BRD4
SCHEMBL24578981 0.81 MEN1 (0.44) SMPD1BRD4NPC1RAB9AMEN1
SCHEMBL17726575 0.81 BRD4 (0.49) SMPD1BRD4NPC1RAB9AGABRA5
SCHEMBL17726200 0.80 SMPD1 (0.53) SMPD1MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9688644-B2 Synthesis of Tetracyclines and intermediates thereto PRESIDENT AND FELLOWS OF HARVARD COLLEGE (US) 2017-06-27 US disclosed
US-9688644-B2 Synthesis of Tetracyclines and intermediates thereto PRESIDENT AND FELLOWS OF HARVARD COLLEGE (US) 2017-06-27 US disclosed
US-20160002183-A1 SYNTHESIS OF TETRACYCLINES AND INTERMEDIATES THERETO PRESIDENT AND FELLOWS OF HARVARD COLLEGE (US) 2016-01-07 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20160002183-A1 SYNTHESIS OF TETRACYCLINES AND INTERMEDIATES THERETO TECR, TAOK1, TET1 SMPD1 4740/4885BRD4 2385/4885NPC1 2850/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.