SCHEMBL1742086

SCHEMBL1742086

O=C(NC1CC1)c1ccc(N2CCN(Cc3cnc4c(c3)NC(=O)[C@@H]3CCCCN43)CC2)c(Cl)c1.O=C1Nc2cc(CO)cnc2N2CCCC[C@@H]12

nearest known ligand 0.57

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 17/20 0.57
TNK1 Q13470 3/20 0.48
NTRK1 P04629 1/20 0.46
KDM4E B2RXH2 1/20 0.43
MEN1 O00255 1/20 0.43
ALDH1A1 P00352 1/20 0.43
MAPT P10636 1/20 0.43
HPGD P15428 1/20 0.43
ALOX15 P16050 1/20 0.43
KMT2A Q03164 1/20 0.43
HSD17B10 Q99714 1/20 0.43
TNK2 Q07912 2/20 0.41
PARP2 Q9UGN5 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL709688 0.97 PARP1 (0.60) PARP1TNK1NTRK1KDM4EMEN1
SCHEMBL709469 0.95 PARP1 (0.61) PARP1TNK1NTRK1KDM4EMEN1
SCHEMBL1738902 0.92 PARP1 (0.60) PARP1TNK1NTRK1TNK2
SCHEMBL1742000 0.92 PARP1 (0.49) PARP1TNK1NTRK1KDM4EMEN1
SCHEMBL716551 0.89 PARP1 (0.51) PARP1TNK1NTRK1KDM4EMEN1
SCHEMBL708332 0.89 PARP1 (0.63) PARP1TNK1NTRK1TNK2
SCHEMBL707608 0.89 PARP1 (0.59) PARP1TNK1NTRK1KDM4EMEN1
SCHEMBL1742046 0.88 PARP1 (0.48) PARP1NTRK1KDM4EMEN1ALDH1A1
SCHEMBL1741938 0.88 PARP1 (0.55) PARP1KDM4EMEN1ALDH1A1MAPT
SCHEMBL708165 0.87 PARP1 (0.61) PARP1TNK1NTRK1KDM4EMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2389379-A1 Poly (ADP-Ribose) Polymerase (PARP) Inhibitors Takeda Pharmaceutical Company Limited (JP) 2011-11-30 EP disclosed