SCHEMBL17424939

SCHEMBL17424939

Cc1ccc(F)cc1C[C@H](CI)Nc1cc[nH]c(=O)c1-c1nc2cc3c(cc2[nH]1)CNC3=O

nearest known ligand 0.50

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
NTRK1 P04629 9/20 0.50
ACVRL1 P37023 9/20 0.50
RET P07949 4/20 0.50
ROS1 P08922 4/20 0.50
MET P08581 2/20 0.50
NTRK3 Q16288 2/20 0.43
NTRK2 Q16620 2/20 0.43
IGF1R P08069 11/20 0.42
CYP1A2 P05177 3/20 0.42
CYP3A4 P08684 3/20 0.42
CYP2C9 P11712 3/20 0.42
CYP2C19 P33261 3/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3459244 0.90 NTRK1 (0.60) NTRK1ACVRL1RETROS1MET
SCHEMBL441092 0.90 NTRK1 (0.60) NTRK1ACVRL1RETROS1MET
SCHEMBL16440373 0.87 NTRK1 (0.60) NTRK1ACVRL1RETROS1MET
SCHEMBL469150 0.87 NTRK1 (0.60) NTRK1ACVRL1RETROS1MET
SCHEMBL469163 0.87 NTRK1 (0.60) NTRK1ACVRL1RETROS1MET
SCHEMBL439732 0.83 NTRK1 (0.69) NTRK1ACVRL1RETROS1MET
SCHEMBL16437782 0.83 NTRK1 (0.69) NTRK1ACVRL1RETROS1MET
SCHEMBL441648 0.79 NTRK1 (0.61) NTRK1ACVRL1RETROS1MET
SCHEMBL441500 0.77 NTRK1 (0.71) NTRK1ACVRL1RETROS1MET
SCHEMBL441109 0.77 NTRK1 (0.68) NTRK1ACVRL1RETROS1MET

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2966076-A1 NOVEL TYROSINE KINASE INHIBITORS ChemBridge Corporation (US) 2016-01-13 EP disclosed