SCHEMBL17484240

SCHEMBL17484240

CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCC(N5CCCC5)CC4)cn3)nc2n(C2CCCC2)c1=O

nearest known ligand 0.88

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CDK4 P11802 20/20 0.88
CCND1 P24385 14/20 0.88
CCND3 P30281 12/20 0.88
CCND2 P30279 11/20 0.88
CDK6 Q00534 7/20 0.81
CCNA2 P20248 4/20 0.81
CDK2 P24941 4/20 0.81
CDK9 P50750 2/20 0.81
CCNA1 P78396 2/20 0.81
CHEK1 O14757 1/20 0.81
DAPK3 O43293 1/20 0.81
CCNT1 O60563 1/20 0.81
CCNT2 O60583 1/20 0.81
ROCK2 O75116 1/20 0.81
STK16 O75716 1/20 0.81
CCNK O75909 1/20 0.81
PDE5A O76074 1/20 0.81
PRKD3 O94806 1/20 0.81
CCNB2 O95067 1/20 0.81
ABCB11 O95342 1/20 0.81

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17484245 0.99 CDK4 (0.89) CDK4CCND1CCND3CCND2CDK6
SCHEMBL17484294 0.98 CDK4 (0.85) CDK4CCND1CCND3CCND2CDK6
SCHEMBL17484239 0.95 CDK4 (0.90) CDK4CCND1CCND3CCND2CDK6
SCHEMBL29507588 0.94 CDK4 (0.98) CDK4CCND1CCND3CCND2CDK6
SCHEMBL4832978 0.94 CDK4 (0.98) CDK4CCND1CCND3CCND2CDK6
SCHEMBL17484269 0.94 CDK4 (0.80) CDK4CCND1CCND3CCND2CDK6
SCHEMBL17479144 0.94 CDK4 (0.90) CDK4CCND1CCND3CCND2CDK6
SCHEMBL31607866 0.94 CDK4 (0.90) CDK4CCND1CCND3CCND2CDK6
SCHEMBL4833113 0.94 CDK4 (1.00) CDK4CCND1CCND3CCND2CDK6
SCHEMBL4832769 0.94 CDK4 (1.00) CDK4CCND1CCND3CCND2CDK6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2016015597-A1 COMPOUNDS AS CDK SMALL-MOLECULE INHIBITORS AND USES THEREOF SUNSHINE LAKE PHARMA CO., LTD. (CN) 2016-02-04 WO disclosed