SCHEMBL17485367

SCHEMBL17485367

Cc1nc2c(F)cc(-c3nc(Nc4ncc(C(=O)N5CC(O)C5)cn4)ncc3F)cc2n1C(C)C

nearest known ligand 0.62

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CDK4 P11802 20/20 0.62
CDK6 Q00534 16/20 0.62
CCND3 P30281 10/20 0.62
CCND1 P24385 9/20 0.62
CDK2 P24941 8/20 0.58
CDK1 P06493 4/20 0.58
CCNB1 P14635 4/20 0.58
CCNA2 P20248 1/20 0.58
KDR P35968 1/20 0.58
CCNE1 P24864 3/20 0.55
HDAC3 O15379 1/20 0.55
HDAC1 Q13547 1/20 0.55
HDAC10 Q969S8 1/20 0.55
HDAC6 Q9UBN7 1/20 0.55
CDK7 P50613 1/20 0.55
CDK9 P50750 1/20 0.55

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17477193 0.91 CDK4 (0.62) CDK4CDK6CCND3CCND1CDK2
SCHEMBL17485357 0.88 CDK4 (0.63) CDK4CDK6CCND3CCND1CDK2
SCHEMBL17485352 0.87 CDK4 (0.59) CDK4CDK6CCND3CCND1CDK2
SCHEMBL17485363 0.86 CDK4 (0.61) CDK4CDK6CCND3CCND1CDK2
SCHEMBL17485420 0.86 CDK4 (0.66) CDK4CDK6CCND3CCND1CDK2
SCHEMBL17485368 0.86 CDK4 (0.62) CDK4CDK6CCND3CCND1CDK2
SCHEMBL17485365 0.85 CDK4 (0.57) CDK4CDK6CCND3CCND1CDK2
SCHEMBL17488630 0.85 CDK4 (0.61) CDK4CDK6CCND3CCND1CDK2
SCHEMBL17488699 0.85 CDK4 (0.61) CDK4CDK6CCND3CCND1CDK2
SCHEMBL17485354 0.84 CDK4 (0.65) CDK4CDK6CCND3CCND1CDK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2016015604-A1 COMPOUNDS AS CDK SMALL-MOLECULE INHIBITORS AND USES THEREOF SUNSHINE LAKE PHARMA CO., LTD. (CN) 2016-02-04 WO disclosed