SCHEMBL17485387

SCHEMBL17485387

CCN1CCc2cc(Nc3ncc(F)c(-c4cc(F)c5nc(C)n(C(C)C)c5c4)n3)ncc2C1

nearest known ligand 0.79

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CDK4 P11802 20/20 0.79
CDK1 P06493 12/20 0.79
CCNB1 P14635 11/20 0.79
CCNE1 P24864 11/20 0.79
CDK6 Q00534 14/20 0.68
CDK2 P24941 13/20 0.68
CDK9 P50750 5/20 0.68
CDK7 P50613 4/20 0.68
CCND3 P30281 4/20 0.68
CCNT1 O60563 3/20 0.68
CCNA2 P20248 3/20 0.68
EGFR P00533 2/20 0.68
NTRK1 P04629 2/20 0.68
BRAF P15056 2/20 0.68
KDR P35968 2/20 0.68
MAPK8 P45983 2/20 0.68
CCNH P51946 2/20 0.68
MNAT1 P51948 2/20 0.68
MAPK10 P53779 2/20 0.68
CDK5 Q00535 2/20 0.68

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18289048 0.88 CDK4 (1.00) CDK4CDK1CCNB1CCNE1CDK6
SCHEMBL17477262 0.88 CDK4 (1.00) CDK4CDK1CCNB1CCNE1CDK6
SCHEMBL22003548 0.84 CDK4 (0.73) CDK4CDK1CCNB1CCNE1CDK6
SCHEMBL17485309 0.82 CDK4 (0.79) CDK4CDK1CCNB1CCNE1CDK6
SCHEMBL17485373 0.82 CDK4 (0.80) CDK4CDK1CCNB1CCNE1CDK6
SCHEMBL21795786 0.82 CDK4 (0.74) CDK4CDK1CCNB1CCNE1CDK6
SCHEMBL22003440 0.82 CDK4 (0.71) CDK4CDK1CCNB1CCNE1CDK6
SCHEMBL17485323 0.82 CDK4 (0.74) CDK4CDK1CCNB1CCNE1CDK6
SCHEMBL17485406 0.82 CDK4 (0.79) CDK4CDK1CCNB1CCNE1CDK6
SCHEMBL17485337 0.82 CDK4 (0.79) CDK4CDK1CCNB1CCNE1CDK6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2016015604-A1 COMPOUNDS AS CDK SMALL-MOLECULE INHIBITORS AND USES THEREOF SUNSHINE LAKE PHARMA CO., LTD. (CN) 2016-02-04 WO disclosed