SCHEMBL17488690

SCHEMBL17488690

Cc1nc2c(F)cc(-c3nc(Nc4ccc(N5CC6CC5CN6C)cn4)ncc3F)cc2n1C(C)C

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CDK4 P11802 19/20 0.59
CDK6 Q00534 14/20 0.59
CDK2 P24941 13/20 0.59
CDK1 P06493 13/20 0.59
CCNB1 P14635 10/20 0.59
CCNE1 P24864 10/20 0.59
CDK9 P50750 7/20 0.59
CDK7 P50613 6/20 0.59
CCND3 P30281 4/20 0.59
CCNA2 P20248 3/20 0.59
EGFR P00533 3/20 0.59
CCNT1 O60563 3/20 0.59
NTRK1 P04629 2/20 0.59
BRAF P15056 2/20 0.59
KDR P35968 2/20 0.59
MAPK8 P45983 2/20 0.59
CCNH P51946 2/20 0.59
MNAT1 P51948 2/20 0.59
MAPK10 P53779 2/20 0.59
CDK5 Q00535 2/20 0.59

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17489094 0.90 CDK4 (0.63) CDK4CDK6CDK2CDK1CCNB1
SCHEMBL17489232 0.87 CDK4 (0.62) CDK4CDK6CDK2CDK1CCNB1
SCHEMBL17488691 0.86 CDK4 (0.69) CDK4CDK6CDK2CDK1CCNB1
SCHEMBL17488689 0.85 CDK4 (0.56) CDK4CDK6CDK2CDK1CCNB1
SCHEMBL17488730 0.84 CDK4 (0.62) CDK4CDK6CDK2CDK1CCNB1
SCHEMBL17477188 0.83 CDK4 (0.63) CDK4CDK6CDK2CDK1CCNB1
SCHEMBL17488687 0.83 CDK4 (0.62) CDK4CDK6CDK2CDK1CCNB1
SCHEMBL17488768 0.83 CDK4 (0.62) CDK4CDK6CDK2CDK1CCNB1
SCHEMBL17489234 0.83 EGFR (0.63) CDK4CDK6CDK2CDK1CCNB1
SCHEMBL17477181 0.82 CDK4 (0.60) CDK4CDK6CDK2CDK1CCNB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2016015605-A1 COMPOUNDS AS CDK SMALL-MOLECULE INHIBITORS AND USES THEREOF SUNSHINE LAKE PHARMA CO., LTD. (CN) 2016-02-04 WO disclosed