SCHEMBL17488753

SCHEMBL17488753

COC(=O)N[C@@H]1CCN(Cc2ccc(Nc3ncc(F)c(-c4cc(F)c5nc(C)n(C(C)C)c5c4)n3)nc2)C1

nearest known ligand 0.69

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CDK4 P11802 20/20 0.69
CDK6 Q00534 16/20 0.69
CDK2 P24941 12/20 0.69
CDK1 P06493 9/20 0.69
CCNB1 P14635 7/20 0.69
CCNE1 P24864 7/20 0.69
CCND3 P30281 6/20 0.69
CDK9 P50750 4/20 0.69
CCNA2 P20248 3/20 0.69
CDK7 P50613 3/20 0.69
CCND1 P24385 3/20 0.69
CCNT1 O60563 2/20 0.69
CIT O14578 1/20 0.69
GAK O14976 1/20 0.69
DYRK3 O43781 1/20 0.69
STK16 O75716 1/20 0.69
CCNK O75909 1/20 0.69
STK10 O94804 1/20 0.69
PRKD3 O94806 1/20 0.69
ABCB11 O95342 1/20 0.69

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17489055 0.90 CDK4 (0.76) CDK4CDK6CDK2CDK1CCNB1
SCHEMBL17489284 0.90 CDK4 (0.76) CDK4CDK6CDK2CDK1CCNB1
SCHEMBL17489053 0.90 CDK4 (0.76) CDK4CDK6CDK2CDK1CCNB1
SCHEMBL17488670 0.89 CDK4 (0.71) CDK4CDK6CDK2CDK1CCNB1
SCHEMBL17488671 0.89 CDK4 (0.71) CDK4CDK6CDK2CDK1CCNB1
SCHEMBL17488736 0.88 CDK4 (0.58) CDK4CDK6CDK2CDK1CCNB1
SCHEMBL17488747 0.88 CDK4 (0.77) CDK4CDK6CDK2CDK1CCNB1
SCHEMBL17488714 0.86 CDK4 (0.80) CDK4CDK6CDK2CDK1CCNB1
SCHEMBL17488700 0.86 CDK4 (0.82) CDK4CDK6CDK2CDK1CCNB1
SCHEMBL17489166 0.86 CDK4 (0.58) CDK4CDK6CDK2CDK1CCNB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2016015605-A1 COMPOUNDS AS CDK SMALL-MOLECULE INHIBITORS AND USES THEREOF SUNSHINE LAKE PHARMA CO., LTD. (CN) 2016-02-04 WO disclosed