SCHEMBL17495269

SCHEMBL17495269

FC1(F)CCNC1CNc1ncccn1

nearest known ligand 0.37

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.37
GRIN2B Q13224 3/20 0.33
HRH4 Q9H3N8 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19227576 0.84 HCRTR1 (0.35)
SCHEMBL23963612 0.71 NPC1 (0.43)
SCHEMBL23963627 0.70 PCSK9 (0.42) ALDH1A1
SCHEMBL20189218 0.70 GRIN2B (0.40) ALDH1A1GRIN2BHRH4
SCHEMBL20189215 0.70 GRIN2B (0.40) ALDH1A1GRIN2BHRH4
SCHEMBL18296935 0.70 GRIN2B (0.40) ALDH1A1GRIN2BHRH4
Hydrochloric Acid SCHEMBL18280955 0.69 GRIN2B (0.40) ALDH1A1GRIN2BHRH4
Hydrochloric Acid SCHEMBL18281002 0.69 GRIN2B (0.40) ALDH1A1GRIN2BHRH4
SCHEMBL1596808 0.68 IDO1 (0.44)
SCHEMBL24288112 0.68 MAP4K4 (0.35) HRH4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3180332-A1 DIFLUOROPYRROLIDINES AS OREXIN RECEPTOR MODULATORS Eolas Therapeutics Inc. (US) 2017-06-21 EP disclosed
WO-2016025669-A1 DIFLUOROPYRROLIDINES AS OREXIN RECEPTOR MODULATORS EOLAS THERAPEUTICS, INC. (US) 2016-02-18 WO disclosed