SCHEMBL17508161

SCHEMBL17508161

C[C@H](C(=O)O)[C@H](O)CN(C)C(=O)OC(C)(C)C

nearest known ligand 0.34

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
CYP2D6 P10635 1/20 0.33
HTR2C P28335 1/20 0.33
SLC6A4 P31645 1/20 0.33
MEN1 O00255 1/20 0.33
GAA P10253 1/20 0.33
KMT2A Q03164 1/20 0.33
HDAC6 Q9UBN7 2/20 0.32
HDAC1 Q13547 1/20 0.32
HDAC2 Q92769 1/20 0.32
CA1 P00915 1/20 0.30
CA2 P00918 1/20 0.30
CA7 P43166 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15597145 1.00 CYP2D6 (0.33) CYP2D6HTR2CSLC6A4MEN1GAA
SCHEMBL13779828 0.83 CYP2D6 (0.33) CYP2D6HDAC6HDAC1HDAC2CA1
SCHEMBL15597130 0.83 CYP2D6 (0.33) CYP2D6HDAC6HDAC1HDAC2CA1
SCHEMBL17898137 0.82 MEN1 (0.34) HTR2CSLC6A4MEN1GAAKMT2A
SCHEMBL10473405 0.82 MEN1 (0.34) HTR2CSLC6A4MEN1GAAKMT2A
SCHEMBL14750621 0.82 MEN1 (0.34) HTR2CSLC6A4MEN1GAAKMT2A
SCHEMBL23134818 0.82 MAPK1 (0.35) CYP2D6HTR2CSLC6A4HDAC6HDAC1
SCHEMBL20215933 0.82 MAPK1 (0.35) CYP2D6HTR2CSLC6A4HDAC6HDAC1
SCHEMBL22916149 0.81 CA14 (0.33) CYP2D6HDAC6HDAC1HDAC2CA1
SCHEMBL1447140 0.80 HDAC6 (0.36) CYP2D6HTR2CSLC6A4MEN1GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2016019588-A1 OXACAZONE COMPOUNDS TO TREAT CLOSTRIDIUM DIFFICILE THE BROAD INSTITUTE, INC. (US) 2016-02-11 WO disclosed