SCHEMBL17516239

SCHEMBL17516239

O=C1c2ccccc2C(=O)N1OI

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GAA P10253 1/20 0.52
ALDH1A1 P00352 6/20 0.48
KMT2A Q03164 4/20 0.48
MAPT P10636 4/20 0.48
KDM4E B2RXH2 3/20 0.48
HPGD P15428 3/20 0.48
CYP1A2 P05177 4/20 0.44
MEN1 O00255 3/20 0.44
VDR P11473 1/20 0.44
CYP2C9 P11712 1/20 0.44
POLB P06746 1/20 0.43
CASP3 P42574 1/20 0.41
HTT P42858 2/20 0.41
CYP3A4 P08684 1/20 0.41
XBP1 P17861 1/20 0.41
CYP2C19 P33261 1/20 0.41
NPSR1 Q6W5P4 1/20 0.41
F2 P00734 1/20 0.41
LMNA P02545 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20768726 0.79 GAA (0.56) GAAALDH1A1KMT2AMAPTKDM4E
SCHEMBL262472 0.79 GAA (0.56) GAAALDH1A1KMT2AMAPTKDM4E
SCHEMBL3359433 0.77 GAA (0.54) GAAALDH1A1KMT2AMAPTKDM4E
SCHEMBL3863655 0.75 GAA (0.52) GAAALDH1A1KMT2AMAPTKDM4E
SCHEMBL798345 0.75 GAA (0.52) GAAALDH1A1KMT2AMAPTKDM4E
SCHEMBL14159314 0.75 GAA (0.52) GAAALDH1A1KMT2AMAPTKDM4E
SCHEMBL12963641 0.75 GAA (0.52) GAAALDH1A1KMT2AMAPTKDM4E
SCHEMBL19341881 0.75 GAA (0.52) GAAALDH1A1KMT2AMAPTKDM4E
SCHEMBL13286163 0.75 GAA (0.52) GAAALDH1A1KMT2AMAPTKDM4E
SCHEMBL13545621 0.75 GAA (0.69) GAAALDH1A1KMT2AMAPTKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3694836-B1 PROCESS FOR PREPARING INTERMEDIATE OF ANTI-TUMOR DRUG NIRAPARIB AND INTERMEDIATE THEREOF ZAI LAB SHANGHAI CO LTD (CN) 2022-06-15 EP disclosed
WO-2016020404-A1 PROCESS FOR THE RESOLUTION OF (R,S)-DIAZEPANE AND DIAZEPANONE DERIVATIVES SANDOZ AG (CH) 2016-02-11 WO disclosed
WO-2016020405-A1 NOVEL ROUTES OF SYNTHESIS FOR THE PREPARATION OF SUVOREXANT SANDOZ AG (CH) 2016-02-11 WO disclosed
WO-2016020403-A1 PREPARATION OF A BENZOIC ACID DERIVATIVE AND ITS USE FOR THE PREPARATION OF SUVOREXANT SANDOZ AG (CH) 2016-02-11 WO disclosed