SCHEMBL17546397

SCHEMBL17546397

Cc1csc(Cl)c1C(=O)NCc1ccc2c(c1)OCO2

nearest known ligand 0.64

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ALDH2 P05091 1/20 0.64
TP53 P04637 1/20 0.60
CRHBP P24387 1/20 0.60
RECQL P46063 1/20 0.60
CRHR2 Q13324 1/20 0.60
NPC1 O15118 1/20 0.60
TDP1 Q9NUW8 1/20 0.59
LMNA P02545 2/20 0.58
KDM4E B2RXH2 1/20 0.58
HPGD P15428 3/20 0.57
L3MBTL1 Q9Y468 1/20 0.56
MAPK1 P28482 2/20 0.56
MEN1 O00255 2/20 0.56
KMT2A Q03164 2/20 0.56
TSHR P16473 2/20 0.56
MMP13 P45452 1/20 0.55
SMN1; SMN2 Q16637 1/20 0.54
ALDH1A1 P00352 1/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10107725 0.88 ALDH2 (0.70) ALDH2TP53CRHBPRECQLCRHR2
SCHEMBL16994124 0.81 ALDH2 (0.77) ALDH2TP53CRHBPRECQLCRHR2
SCHEMBL10107753 0.81 ALDH2 (0.73) ALDH2TP53CRHBPRECQLCRHR2
SCHEMBL10107747 0.78 ALDH2 (0.81) ALDH2TP53CRHBPRECQLCRHR2
SCHEMBL503808 0.78 ALDH2 (1.00) ALDH2TP53CRHBPRECQLCRHR2
SCHEMBL16864898 0.78 TP53 (0.64) ALDH2TP53CRHBPRECQLCRHR2
SCHEMBL16864899 0.77 ALDH2 (0.64) ALDH2TP53CRHBPRECQLCRHR2
SCHEMBL16864900 0.77 ALDH2 (0.74) ALDH2TP53CRHBPRECQLCRHR2
SCHEMBL13435809 0.77 TP53 (0.62) ALDH2TP53CRHBPRECQLCRHR2
SCHEMBL13435819 0.76 ALDH2 (0.69) ALDH2TP53CRHBPRECQLCRHR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9315484-B2 Mitochondrial aldehyde dehydrogenase-2 modulators and methods of use thereof The Board of Trustees—Leland Stanford Junior University (US) 2016-04-19 US disclosed
US-9273025-B2 2016-03-01 US disclosed