Cyclosporine

Cyclosporine

SCHEMBL17555

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nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

PPIA

The experimentally established mechanism targets of Cyclosporine. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PPIA known ✓ P62937 5/20 1.00
ABCB1 P08183 13/20 1.00
PPP3CA Q08209 3/20 1.00
FKBP1B P68106 2/20 1.00
MEN1 O00255 1/20 1.00
NPC1 O15118 1/20 1.00
ABCC3 O15438 1/20 1.00
GMNN O75496 1/20 1.00
USP2 O75604 1/20 1.00
SLCO2B1 O94956 1/20 1.00
ABCB11 O95342 1/20 1.00
LMNA P02545 1/20 1.00
POLB P06746 1/20 1.00
CYP3A4 P08684 1/20 1.00
MAPT P10636 1/20 1.00
RARB P10826 1/20 1.00
CYP2C9 P11712 1/20 1.00
CYP3A5 P20815 1/20 1.00
TACR2 P21452 1/20 1.00
PPIB P23284 1/20 1.00

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Cyclosporine SCHEMBL21170318 1.00 ABCB1 (1.00) ABCB1PPIAPPP3CAFKBP1BMEN1
SCHEMBL23382247 1.00 ABCB1 (1.00) ABCB1PPIAPPP3CAFKBP1BMEN1
Cyclosporine SCHEMBL24239446 1.00 ABCB1 (1.00) ABCB1PPIAPPP3CAFKBP1BMEN1
Cyclosporine SCHEMBL24224445 1.00 ABCB1 (1.00) ABCB1PPIAPPP3CAFKBP1BMEN1
Cyclosporine SCHEMBL25083206 1.00 ABCB1 (1.00) ABCB1PPIAPPP3CAFKBP1BMEN1
Cyclosporine SCHEMBL24239035 1.00 ABCB1 (1.00) ABCB1PPIAPPP3CAFKBP1BMEN1
Cyclosporine SCHEMBL23192320 1.00 ABCB1 (1.00) ABCB1PPIAPPP3CAFKBP1BMEN1
SCHEMBL23110210 1.00 ABCB1 (1.00) ABCB1PPIAPPP3CAFKBP1BMEN1
Cyclosporine SCHEMBL24239036 1.00 ABCB1 (1.00) ABCB1PPIAPPP3CAFKBP1BMEN1
Cyclosporine SCHEMBL23192319 1.00 ABCB1 (1.00) ABCB1PPIAPPP3CAFKBP1BMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Appears in 31454 patents — a generic fragment claimed broadly, so it's down-weighted as IP noise. Top by claim status then date:

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20260139860-A1 PRODUCTS OF MANUFACTURE FOR THE TREATMENT, PREVENTION AND AMELIORATION OF MICROBIAL INFECTIONS CENTRE FOR DIGESTIVE DISEASES (AU) 2026-05-21 US claimed
WO-2026107085-A1 METHODS OF TREATING LUPUS WITH CD19-CD20 DUAL CAR-T CELLS GENENTECH, INC. (US) 2026-05-21 WO claimed
US-20260137558-A1 OPHTHALMIC DEVICE Able Tx Ltd. (IL) 2026-05-21 US claimed
US-20260124148-A1 POLYPEPTIDE FORMULATIONS FOR ORAL DELIVERY BHAMIS RES LABORATORY PVT LTD (IN) 2026-05-07 US claimed
US-20260125770-A1 INFLAMMATORY DISORDER IN A FELIDAE MARS, INCORPORATED (US) 2026-05-07 US claimed
EP-4255391-B1 LUMINOL FOR USE IN THE TREATMENT OF SEQUELAE OF A SARS-COV-2 INFECTION METRIOPHARM AG (CH) 2026-05-06 EP claimed
EP-4736841-A1 A MUCOADHESIVE LAYER FOR BUCCAL ADMINISTRATION OF AN ACTIVE PHARMACEUTICAL INGREDIENT IQ medical GmbH (DE) 2026-05-06 EP claimed
US-20260108619-A1 CONJUGATION LINKERS, CELL BINDING MOLECULE-DRUG CONJUGATES CONTAINING THE LINKERS, METHODS OF MAKING AND USES SUCH CONJUGATES WITH THE LINKERS HANGZHOU DAC BIOTECH CO., LTD. (CN) 2026-04-23 US claimed
US-20260103532-A1 PHARMACEUTICAL COMPOSITIONS OF HUMANIZED ANTI-CD40 ANTIBODIES AND USES THEREOF KINIKSA PHARMACEUTICALS GMBH (CH) 2026-04-16 US claimed
US-20260102373-A1 LYMPH DIRECTING PRODRUGS MONASH UNIVERSITY (AU) 2026-04-16 US claimed
EP-0561772-A1 A new pharmaceutical use of fusidic acid and derivatives thereof BENDTZEN, Klaus (DK) 1993-09-29 EP claimed
EP-0296122-B1 CYCLOSPORINS AND THEIR USE AS PHARMACEUTICALS SANDOZ AG (CH) 1993-09-29 EP claimed
WO-1993017039-A1 ISO-CYCLOSPORIN SALTS SANDOZ LTD. (CH) 1993-09-02 WO claimed
EP-0539319-A2 Pharmaceutical cyclosporin composition SANDOZ LTD. (CH) 1993-04-28 EP claimed
EP-0504760-A1 Ciclosporin form for pulmonary administration SANDOZ LTD. (CH) 1992-09-23 EP claimed
CN-1053010-A PHARMACEUTICAL PREPARATION PUETTER MEDICE CHEM PHARM (DE) 1991-07-17 CN claimed
CN-1051503-A Disease and treatment of diseases NORPHARMCO INC (CA) 1991-05-22 CN claimed
EP-0414632-A2 Cyclosporin derivatives SANDOZ LTD. (CH) 1991-02-27 EP claimed
WO-1990004398-A1 A NEW PHARMACEUTICAL USE OF FUSIDIC ACID AND DERIVATIVES THEREOF BENDTZEN KLAUS (DK) 1990-05-03 WO claimed
EP-0296122-A2 Cyclosporins and their use as pharmaceuticals SANDOZ AG (CH) 1988-12-21 EP claimed