SCHEMBL17558388

SCHEMBL17558388

CC1(C)C(=O)N(c2ccc(SC(F)(F)F)cc2)C(=O)N1Cc1c[c]nc(Cl)c1

nearest known ligand 0.73

Predicted protein targets (top 1)

geneUniProtsupporting neighboursconfidence
IGF1R P08069 19/20 0.73

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2943071 0.87 IGF1R (0.80) IGF1R
SCHEMBL2939981 0.84 IGF1R (1.00) IGF1R
SCHEMBL4851290 0.83 IGF1R (0.76) IGF1R
SCHEMBL2941768 0.83 IGF1R (0.73) IGF1R
SCHEMBL1130587 0.81 IGF1R (1.00) IGF1R
SCHEMBL2941767 0.80 IGF1R (0.76) IGF1R
SCHEMBL13039126 0.79 IGF1R (0.72) IGF1R
SCHEMBL2991808 0.78 IGF1R (0.75) IGF1R
SCHEMBL3728553 0.78 IGF1R (0.63) IGF1R
SCHEMBL2941196 0.77 IGF1R (0.81) IGF1R

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3188729-A1 CYCLIC UREA COMPOUNDS AS TROPOMYOSIN-RELATED KINASE (TRK) INHIBITORS Genzyme Corporation (US) 2017-07-12 EP disclosed
WO-2016036796-A1 CYCLIC UREA COMPOUNDS AS TROPOMYOSIN-RELATED KINASE (TRK) INHIBITORS GENZYME CORPORATION (US) 2016-03-10 WO disclosed