SCHEMBL17595149

SCHEMBL17595149

CCc1cc(C(=O)OC(=O)C(F)(F)F)c(=O)[nH]c1-c1ccc(N2CCC(N(C)C)C2)cc1

nearest known ligand 0.51

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 2/20 0.51
MCHR1 Q99705 13/20 0.40
WDR5 P61964 1/20 0.36
NOTUM Q6P988 1/20 0.35
TLR9 Q9NR96 2/20 0.34
TLR8 Q9NR97 2/20 0.34
TLR7 Q9NYK1 2/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14741135 1.00 KCNH2 (0.51) KCNH2MCHR1WDR5NOTUMTLR9
SCHEMBL14745538 0.92 KCNH2 (0.42) KCNH2MCHR1WDR5NOTUM
SCHEMBL14741004 0.88 KCNH2 (0.38) KCNH2NOTUM
SCHEMBL14745225 0.88 PRKD3 (0.44) KCNH2NOTUM
Trifluoroacetic Acid SCHEMBL17595148 0.87 KCNH2 (0.53) KCNH2MCHR1WDR5
Trifluoroacetic Acid SCHEMBL14741133 0.87 KCNH2 (0.53) KCNH2MCHR1WDR5
SCHEMBL14744736 0.86 TOP1 (0.39) KCNH2
SCHEMBL14758835 0.85 KCNH2 (0.57) KCNH2MCHR1WDR5
SCHEMBL14745687 0.85 KCNH2 (0.57) KCNH2MCHR1WDR5
SCHEMBL14758820 0.85 KCNH2 (0.57) KCNH2MCHR1WDR5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2016039936-A2 MONOCYCLIC SUBSTITUTED 2-PYRIDINONE ANTIBACTERIAL COMPOUNDS PTC THERAPEUTICS, INC. (US) 2016-03-17 WO claimed