SCHEMBL17609167

SCHEMBL17609167

CN(Cc1ccccc1)c1cccc(Oc2ncc3ccncc3n2)c1

nearest known ligand 0.60

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
KDM4C Q9H3R0 4/20 0.60
GRM2 Q14416 3/20 0.42
DHFR P00374 1/20 0.39
CHRNB2 P17787 1/20 0.38
CHRNA4 P43681 1/20 0.38
IP6K1 Q92551 1/20 0.36
USP2 O75604 1/20 0.36
CYP1A2 P05177 1/20 0.36
CYP3A4 P08684 1/20 0.36
CYP2C9 P11712 1/20 0.36
MAPK1 P28482 1/20 0.36
CYP2C19 P33261 1/20 0.36
CLK4 Q9HAZ1 1/20 0.36
CETP P11597 1/20 0.36
F2 P00734 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30139682 1.00 KDM4C (0.60) KDM4CGRM2DHFRCHRNB2CHRNA4
SCHEMBL17609132 0.88 KDM4C (0.58) KDM4CGRM2DHFRIP6K1USP2
SCHEMBL17609100 0.85 KDM4C (0.56) KDM4CGRM2
SCHEMBL30139683 0.85 KDM4C (0.56) KDM4CGRM2
SCHEMBL17602152 0.82 KDM4C (0.65) KDM4CGRM2DHFRCETP
SCHEMBL29542623 0.82 KDM4C (0.65) KDM4CGRM2DHFRCETP
SCHEMBL17609163 0.77 KDM4C (0.54) KDM4C
SCHEMBL30139680 0.77 KDM4C (0.54) KDM4C
SCHEMBL17602155 0.73 KDM4C (0.50) KDM4CGRM2DHFRCHRNB2CHRNA4
SCHEMBL17602292 0.73 KDM4C (0.58) KDM4C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20230117519-A1 HISTONE DEMETHYLASE INHIBITORS CELGENE QUANTICEL RESEARCH, INC. (US) 2023-04-20 US disclosed
US-11535616-B2 Histone demethylase inhibitors CELGENE QUANTICEL RESEARCH, INC (US) 2022-12-27 US disclosed
US-20210009585-A1 HISTONE DEMETHYLASE INHIBITORS CELGENE QUANTICEL RESEARCH, INC. (US) 2021-01-14 US disclosed
US-10815234-B2 Histone demethylase inhibitors CELGENE QUANTICEL RESEARCH, INC. (US) 2020-10-27 US disclosed
US-20200199122-A1 HISTONE DEMETHYLASE INHIBITORS CELGENE QUANTICEL RESEARCH, INC. (US) 2020-06-25 US disclosed
US-10611763-B2 Histone demethylase inhibitors CELGENE QUANTICEL RESEARCH, INC. (US) 2020-04-07 US disclosed
US-20190023704-A1 HISTONE DEMETHYLASE INHIBITORS CELGENE QUANTICEL RESEARCH, INC. (US) 2019-01-24 US disclosed
EP-3193601-A1 HISTONE DEMETHYLASE INHIBITORS Celgene Quanticel Research, Inc. (US) 2017-07-26 EP disclosed
WO-2016044429-A1 HISTONE DEMETHYLASE INHIBITORS Quanticel Pharmaceuticals, Inc. (US) 2016-03-24 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (7 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-10611763-B2 Histone demethylase inhibitors KDM1B, KDM1A, KDM5C KDM4C 9/4885GRM2 2310/4885DHFR 319/4885
US-11535616-B2 Histone demethylase inhibitors KDM1B, KDM1A, KDM5C KDM4C 9/4885GRM2 2310/4885DHFR 319/4885
US-20190023704-A1 HISTONE DEMETHYLASE INHIBITORS KDM1B, KDM1A, KDM5C KDM4C 9/4885GRM2 2310/4885DHFR 319/4885
US-20200199122-A1 HISTONE DEMETHYLASE INHIBITORS KDM1B, KDM1A, KDM5C KDM4C 9/4885GRM2 2310/4885DHFR 319/4885
US-20230117519-A1 HISTONE DEMETHYLASE INHIBITORS KDM1B, KDM1A, KDM5C KDM4C 9/4885GRM2 2310/4885DHFR 319/4885
US-20210009585-A1 HISTONE DEMETHYLASE INHIBITORS KDM1B, KDM1A, KDM5C KDM4C 9/4885GRM2 2310/4885DHFR 319/4885
US-10815234-B2 Histone demethylase inhibitors KDM1B, KDM1A, KDM5C KDM4C 9/4885GRM2 2310/4885DHFR 319/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.