SCHEMBL1761124

SCHEMBL1761124

Cc1cnc(Nc2cncnc2)c(C(=O)Nc2ccc(F)cn2)n1

nearest known ligand 0.66

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
GRM5 P41594 5/20 0.66
PDE10A Q9Y233 14/20 0.52
CYP1A2 P05177 1/20 0.52
CYP2C9 P11712 1/20 0.52
KCNH2 Q12809 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL1761107 0.87 GRM5 (0.66) GRM5PDE10A
SCHEMBL17685489 0.82 GRM5 (0.52) GRM5PDE10ACYP1A2CYP2C9KCNH2
SCHEMBL12595513 0.79 PDE10A (0.59) GRM5PDE10A
Hydrochloric Acid SCHEMBL1761121 0.78 PDE10A (0.58) GRM5PDE10A
Hydrochloric Acid SCHEMBL1385315 0.78 PDE10A (0.50) GRM5PDE10A
SCHEMBL1386262 0.76 PDE10A (0.52) GRM5PDE10A
SCHEMBL2160345 0.75 PDE10A (0.50) PDE10A
Hydrochloric Acid SCHEMBL1383785 0.74 PDE10A (0.55) GRM5PDE10A
Hydrochloric Acid SCHEMBL1383957 0.72 GRM5 (0.63) GRM5
SCHEMBL15663452 0.71 GRM5 (0.52) GRM5PDE10ACYP1A2CYP2C9KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7947685-B2 Pyrazine-2-carboxyamide derivatives HOFFMANN-LA ROCHE INC. (US) 2011-05-24 US disclosed