SCHEMBL17635522

SCHEMBL17635522

CC(=O)c1cccc(C2(C)CCSC(N)=N2)c1

nearest known ligand 0.62

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
BACE1 P56817 20/20 0.62
APP P05067 1/20 0.58
KCNH2 Q12809 1/20 0.57

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10156225 0.90 BACE1 (0.66) BACE1APPKCNH2
SCHEMBL10157601 0.86 BACE1 (0.62) BACE1APPKCNH2
SCHEMBL10155131 0.85 BACE1 (0.80) BACE1APP
SCHEMBL10154574 0.85 BACE1 (0.59) BACE1APPKCNH2
SCHEMBL10157123 0.85 BACE1 (0.59) BACE1APPKCNH2
SCHEMBL10157884 0.85 BACE1 (0.76) BACE1APP
SCHEMBL10154943 0.84 BACE1 (0.55) BACE1APPKCNH2
SCHEMBL15041116 0.84 BACE1 (0.64) BACE1KCNH2
SCHEMBL10154673 0.83 BACE1 (0.64) BACE1APPKCNH2
SCHEMBL10267051 0.83 BACE1 (0.67) BACE1KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2597087-B1 Dihydrooxazine and tetrahydropyrimidine derivatives as BACE 1 inhibitors SHIONOGI & CO (JP) 2016-03-30 EP disclosed