SCHEMBL17635682

SCHEMBL17635682

NN(Cc1ccc(-c2ccccn2)cc1)CC(O)C(Cc1ccccc1)NO

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
UGT1A1 P22309 3/20 0.49
MLNR O43193 1/20 0.49
NR1I2 O75469 1/20 0.49
SLCO2B1 O94956 1/20 0.49
ABCB11 O95342 1/20 0.49
ABCB1 P08183 1/20 0.49
CCKAR P32238 1/20 0.49
OPRK1 P41145 1/20 0.49
GHSR Q92847 1/20 0.49
SLCO1B3 Q9NPD5 1/20 0.49
ABCG2 Q9UNQ0 1/20 0.49
SLCO1B1 Q9Y6L6 1/20 0.49
KCNH2 Q12809 1/20 0.39
DPP4 P27487 1/20 0.37
HCAR2 Q8TDS4 1/20 0.35
MME P08473 1/20 0.35
PPARG P37231 1/20 0.35
TPH1 P17752 1/20 0.34
CETP P11597 1/20 0.34
CA2 P00918 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3553186 0.89 UGT1A1 (0.56) UGT1A1MLNRNR1I2SLCO2B1ABCB11
SCHEMBL3553181 0.89 UGT1A1 (0.56) UGT1A1MLNRNR1I2SLCO2B1ABCB11
SCHEMBL17635757 0.88 CYP2D6 (0.53) UGT1A1MLNRNR1I2SLCO2B1ABCB11
SCHEMBL3393562 0.85 UGT1A1 (0.43) UGT1A1MLNRNR1I2SLCO2B1ABCB11
SCHEMBL2177873 0.85 UGT1A1 (0.43) UGT1A1MLNRNR1I2SLCO2B1ABCB11
SCHEMBL8152590 0.85 UGT1A1 (0.43) UGT1A1MLNRNR1I2SLCO2B1ABCB11
Hydrochloric Acid SCHEMBL1300940 0.84 UGT1A1 (0.43) UGT1A1MLNRNR1I2SLCO2B1ABCB11
Hydrochloric Acid SCHEMBL6156798 0.84 UGT1A1 (0.43) UGT1A1MLNRNR1I2SLCO2B1ABCB11
Hydrochloric Acid SCHEMBL30018372 0.84 UGT1A1 (0.43) UGT1A1MLNRNR1I2SLCO2B1ABCB11
SCHEMBL7907823 0.82 UGT1A1 (0.60) UGT1A1MLNRNR1I2SLCO2B1ABCB11

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2069303-B1 ANTIVIRAL PROTEASE INHIBITORS GILEAD SCIENCES INC (US) 2016-03-30 EP disclosed