SCHEMBL17644202

SCHEMBL17644202

CC(C)(C)OC(=O)N1CCCC1c1ncc(-c2ccc3cc(-c4ccc(-c5cnc(C6CC(C#N)CN6C(=O)O)[nH]5)cc4)ccc3c2)[nH]1

nearest known ligand 0.45

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
PRCP P42785 10/20 0.45
CYP3A4 P08684 3/20 0.43
CYP2C9 P11712 3/20 0.43
NR1I2 O75469 2/20 0.43
KCNH2 Q12809 2/20 0.43
ABCB11 O95342 1/20 0.43
OPRK1 P41145 1/20 0.43
HPGDS O60760 3/20 0.43
CYP1A2 P05177 2/20 0.41
CYP2D6 P10635 1/20 0.41
HCRTR1 O43613 2/20 0.39
HCRTR2 O43614 2/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL204518 0.96 CYP3A4 (0.47) PRCPCYP3A4CYP2C9NR1I2KCNH2
SCHEMBL9980309 0.96 CYP3A4 (0.47) PRCPCYP3A4CYP2C9NR1I2KCNH2
SCHEMBL203107 0.87 CYP3A4 (0.54) PRCPCYP3A4CYP2C9NR1I2KCNH2
SCHEMBL2710848 0.87 CYP3A4 (0.54) PRCPCYP3A4CYP2C9NR1I2KCNH2
SCHEMBL2757500 0.87 CYP3A4 (0.54) PRCPCYP3A4CYP2C9NR1I2KCNH2
SCHEMBL17644210 0.87 PRCP (0.47) PRCPCYP3A4CYP2C9NR1I2KCNH2
SCHEMBL27978753 0.85 PRCP (0.46) PRCPCYP3A4CYP2C9NR1I2KCNH2
SCHEMBL15368504 0.85 CYP2C9 (0.49) PRCPCYP3A4CYP2C9NR1I2KCNH2
SCHEMBL27978669 0.85 PRCP (0.44) PRCPCYP3A4CYP2C9NR1I2KCNH2
SCHEMBL2709400 0.85 PRCP (0.54) PRCPCYP3A4CYP2C9NR1I2KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3626716-A1 ANTIVIRAL COMPOUNDS Gilead Pharmasset LLC (US) 2020-03-25 EP disclosed
EP-3309157-A1 ANTIVIRAL COMPOUNDS Gilead Pharmasset LLC (US) 2018-04-18 EP disclosed
EP-3002281-B1 ANTIVIRAL COMPOUNDS GILEAD PHARMASSET LLC (US) 2017-09-13 EP disclosed
EP-3002281-A1 ANTIVIRAL COMPOUNDS Gilead Pharmasset LLC (US) 2016-04-06 EP disclosed