SCHEMBL17644334

SCHEMBL17644334

Cc1cc(OC(=O)O)nc(N2CC3CN(C(=O)c4c(F)cccc4-n4nccn4)CC3C2)n1

nearest known ligand 0.84

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
HCRTR1 O43613 20/20 0.84
HCRTR2 O43614 20/20 0.84
KCNH2 Q12809 1/20 0.67

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1671265 0.91 HCRTR1 (1.00) HCRTR1HCRTR2
SCHEMBL17644358 0.91 HCRTR1 (0.80) HCRTR1HCRTR2KCNH2
Seltorexant SCHEMBL1671257 0.90 HCRTR1 (1.00) HCRTR1HCRTR2KCNH2
Seltorexant SCHEMBL29614942 0.90 HCRTR1 (1.00) HCRTR1HCRTR2KCNH2
Seltorexant SCHEMBL29711733 0.90 HCRTR1 (1.00) HCRTR1HCRTR2KCNH2
Seltorexant SCHEMBL19341242 0.90 HCRTR1 (1.00) HCRTR1HCRTR2KCNH2
Seltorexant SCHEMBL22018191 0.90 HCRTR1 (1.00) HCRTR1HCRTR2KCNH2
Seltorexant SCHEMBL29577602 0.89 HCRTR1 (0.98) HCRTR1HCRTR2KCNH2
Seltorexant SCHEMBL17270584 0.89 HCRTR1 (0.98) HCRTR1HCRTR2KCNH2
SCHEMBL6924591 0.88 HCRTR1 (0.78) HCRTR1HCRTR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2491038-B1 DISUBSTITUTED OCTAHY - DROPYRROLO [3,4-C]PYRROLES AS OREXIN RECEPTOR MODULATORS JANSSEN PHARMACEUTICA NV (BE) 2016-04-06 EP claimed