SCHEMBL17644580

SCHEMBL17644580

CCOc1cc(C2CN(C=O)CCO2)ccc1Nc1ncc(Br)c(NCCOC)n1

nearest known ligand 0.54

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
LRRK2 Q5S007 10/20 0.54
JAK2 O60674 1/20 0.40
ULK1 O75385 3/20 0.39
EGFR P00533 2/20 0.39
ALK Q9UM73 3/20 0.39
TTK P33981 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17644596 0.95 LRRK2 (0.59) LRRK2JAK2ULK1EGFRALK
SCHEMBL17644531 0.92 LRRK2 (0.60) LRRK2JAK2ULK1EGFRALK
SCHEMBL20537463 0.86 LRRK2 (0.49) LRRK2JAK2ALK
SCHEMBL17644512 0.86 LRRK2 (0.59) LRRK2JAK2EGFRALK
SCHEMBL20537315 0.84 LRRK2 (0.48) LRRK2JAK2ULK1EGFRALK
SCHEMBL17644555 0.84 LRRK2 (0.56) LRRK2JAK2ULK1EGFRALK
SCHEMBL17644572 0.83 LRRK2 (0.62) LRRK2JAK2EGFRALK
SCHEMBL20537296 0.82 LRRK2 (0.58) LRRK2JAK2ULK1EGFRALK
SCHEMBL17644523 0.81 LRRK2 (0.60) LRRK2JAK2ULK1ALK
SCHEMBL17644587 0.81 LRRK2 (0.51) LRRK2JAK2EGFRALK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2576541-B1 AMINOPYRIMIDINE DERIVATIVES AS LRRK2 MODULATORS HOFFMANN LA ROCHE (CH) 2016-04-06 EP claimed