SCHEMBL17656540

SCHEMBL17656540

C=C(C)OC(=O)NCc1cccc(-c2cnc(N3CCN(Cc4ccc(C(=O)OCc5ccccc5)cc4)CC3)nc2)c1

nearest known ligand 0.46

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
FLT1 P17948 2/20 0.46
KDR P35968 2/20 0.46
FLT3 P36888 2/20 0.46
TRPA1 O75762 2/20 0.45
HDAC6 Q9UBN7 1/20 0.41
AOC3 Q16853 5/20 0.40
AURKA O14965 1/20 0.40
BCL2L1 Q07817 1/20 0.40
CHRM3 P20309 2/20 0.39
ROCK2 O75116 1/20 0.39
DRD2 P14416 1/20 0.39
DRD4 P21917 1/20 0.39
DRD3 P35462 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16784890 0.89 FLT1 (0.44) FLT1KDRFLT3TRPA1HDAC6
SCHEMBL17703745 0.86 HDAC6 (0.46) TRPA1HDAC6AOC3BCL2L1DRD2
SCHEMBL17656757 0.84 AOC3 (0.48) HDAC6AOC3BCL2L1DRD2DRD4
SCHEMBL12526352 0.84 AOC3 (0.47) HDAC6AOC3BCL2L1DRD2DRD4
SCHEMBL16784924 0.83 AOC3 (0.45) FLT1KDRFLT3TRPA1HDAC6
SCHEMBL12526638 0.83 AOC3 (0.49) HDAC6AOC3BCL2L1DRD2DRD4
SCHEMBL16785024 0.81 AOC3 (0.48) FLT1KDRFLT3HDAC6AOC3
SCHEMBL17703740 0.74 AOC3 (0.55) AOC3BCL2L1DRD2DRD4DRD3
SCHEMBL16785169 0.73 AOC3 (0.50) HDAC6AOC3BCL2L1DRD2DRD4
SCHEMBL16784922 0.72 AOC3 (0.49) HDAC6AOC3CHRM3ROCK2DRD2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3002278-A1 GUANIDINE COMPOUND Astellas Pharma Inc. (JP) 2016-04-06 EP disclosed