SCHEMBL17675229

SCHEMBL17675229

CCCc1ccnc(NC(=O)c2ccc(Oc3ccnc4ccc(N)cc34)cc2)c1

nearest known ligand 0.62

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
BTK Q06187 16/20 0.62
EGFR P00533 10/20 0.62
TEC P42680 2/20 0.62
TXK P42681 2/20 0.62
BLK P51451 2/20 0.62
BMX P51813 2/20 0.62
ERBB4 Q15303 2/20 0.62
ERBB2 P04626 1/20 0.62
JAK3 P52333 1/20 0.62
NPC1 O15118 1/20 0.44
PKM P14618 1/20 0.44
RAB9A P51151 1/20 0.44
SMN1; SMN2 Q16637 1/20 0.44
MET P08581 1/20 0.42
AXL P30530 1/20 0.42
MERTK Q12866 1/20 0.42
NR3C2 P08235 1/20 0.41
LCK P06239 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17675289 0.93 BTK (0.72) BTKEGFRTECTXKBLK
SCHEMBL17675363 0.87 BTK (0.75) BTKEGFRTECTXKBLK
SCHEMBL17675247 0.86 BTK (0.69) BTKEGFRTECTXKBLK
SCHEMBL17675438 0.85 BTK (0.59) BTKEGFRTECTXKBLK
SCHEMBL17675360 0.84 EGFR (0.87) BTKEGFRTECTXKBLK
SCHEMBL17675235 0.82 BTK (0.73) BTKEGFRTECTXKBLK
SCHEMBL17675205 0.82 BTK (0.58) BTKEGFRTECTXKBLK
SCHEMBL17675216 0.81 BTK (0.54) BTKEGFRTECTXKBLK
SCHEMBL17675250 0.81 BTK (0.78) BTKEGFRTECTXKBLK
SCHEMBL17683767 0.80 BTK (0.77) BTKEGFRTECTXKBLK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2016055982-A1 QUINOLINE AND QUINAZOLINE COMPOUNDS ACERTA PHARMA B.V. (NL) 2016-04-14 WO claimed
WO-2016055982-A1 QUINOLINE AND QUINAZOLINE COMPOUNDS ACERTA PHARMA B.V. (NL) 2016-04-14 WO disclosed