SCHEMBL17675753

SCHEMBL17675753

COc1ccc2c(c1)C(Cc1ccccc1)C(=N)CC2

nearest known ligand 0.50

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 3/20 0.50
SIGMAR1 Q99720 3/20 0.46
HTR1A P08908 1/20 0.43
GRIN1 Q05586 3/20 0.43
GRIN2B Q13224 3/20 0.43
AR P10275 2/20 0.42
KDM1A O60341 2/20 0.42
MAOA P21397 2/20 0.42
MAOB P27338 2/20 0.42
CYP19A1 P11511 1/20 0.41
HTR2C P28335 1/20 0.41
HTR2B P41595 1/20 0.41
CYP24A1 Q07973 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6826968 0.84 HTR2A (0.50) HTR2ASIGMAR1HTR1AGRIN1GRIN2B
SCHEMBL14151721 0.81 HTR2A (0.47) HTR2ASIGMAR1HTR1AGRIN1GRIN2B
SCHEMBL14151720 0.81 HTR2A (0.47) HTR2ASIGMAR1HTR1AGRIN1GRIN2B
SCHEMBL13827955 0.79 GRIN1 (0.45) HTR2ASIGMAR1HTR1AGRIN1GRIN2B
SCHEMBL606089 0.78 HTR2A (0.56) HTR2ASIGMAR1HTR1AARCYP19A1
Bromide SCHEMBL13835350 0.78 HTR2A (0.44) HTR2ASIGMAR1HTR1AGRIN1GRIN2B
SCHEMBL14151107 0.78 HTR2A (0.46) HTR2ASIGMAR1HTR1AARCYP19A1
SCHEMBL13736116 0.76 TACR2 (0.46) HTR2ASIGMAR1HTR1AARMAOA
SCHEMBL3284717 0.74 HTR2A (0.50) HTR2ASIGMAR1GRIN1GRIN2BAR
SCHEMBL10348907 0.74 SLC22A1 (0.63)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9309200-B2 Benzazepine derivatives, pharmaceutical compositions containing them, and their use in therapy AbbVie Deutschland GmbH & Co. KG (DE) 2016-04-12 US disclosed