SCHEMBL17679503

SCHEMBL17679503

CC(C)(C)c1cc(C(C)(C)C)c(ON)cc1NC(=O)c1c[nH]c2ccccc2c1=O

nearest known ligand 0.74

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
CFTR P13569 20/20 0.74
ADORA3 P0DMS8 1/20 0.74
ADRB3 P13945 1/20 0.74
TBXA2R P21731 1/20 0.74
SLC6A2 P23975 1/20 0.74
AGTR1 P30556 1/20 0.74
MC4R P32245 1/20 0.74
PTGS2 P35354 1/20 0.74
SLC6A3 Q01959 1/20 0.74

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL26734614 0.91 CFTR (0.76) CFTRADORA3ADRB3TBXA2RSLC6A2
SCHEMBL26734206 0.90 CFTR (0.74) CFTRADORA3ADRB3TBXA2RSLC6A2
SCHEMBL25874767 0.90 CFTR (0.74) CFTRADORA3ADRB3TBXA2RSLC6A2
SCHEMBL17030124 0.90 CFTR (0.74) CFTRADORA3ADRB3TBXA2RSLC6A2
SCHEMBL6730386 0.89 CFTR (0.73) CFTRADORA3ADRB3TBXA2RSLC6A2
SCHEMBL22872817 0.89 CFTR (0.73) CFTRADORA3ADRB3TBXA2RSLC6A2
SCHEMBL22591867 0.88 CFTR (0.71) CFTRADORA3ADRB3TBXA2RSLC6A2
SCHEMBL19393869 0.88 CFTR (0.71) CFTRADORA3ADRB3TBXA2RSLC6A2
SCHEMBL4174033 0.88 CFTR (0.71) CFTRADORA3ADRB3TBXA2RSLC6A2
SCHEMBL2104014 0.87 CFTR (0.70) CFTRADORA3ADRB3TBXA2RSLC6A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2016057730-A1 CO-CRYSTALS OF MODULATORS OF CYSTIC FIBROSIS TRANSMEMBRANE CONDUCTANCE REGULATOR STROHMEIER MARK (US) 2016-04-14 WO disclosed