SCHEMBL1768048

SCHEMBL1768048

Nc1nc(C(=O)N2Cc3ccccc3C2)c2cc(C3CCC3)ccc2n1

nearest known ligand 0.69

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HSP90AA1 P07900 11/20 0.69
HSP90AB1 P08238 3/20 0.69
EGLN1 Q9GZT9 2/20 0.42
KCNH2 Q12809 2/20 0.38
HRH4 Q9H3N8 2/20 0.38
HRH3 Q9Y5N1 2/20 0.38
NAMPT P43490 1/20 0.38
MMP9 P14780 1/20 0.38
IKBKE Q14164 1/20 0.37
TBK1 Q9UHD2 1/20 0.37
MEN1 O00255 1/20 0.37
ALDH1A1 P00352 1/20 0.37
LMNA P02545 1/20 0.37
TP53 P04637 1/20 0.37
MAPT P10636 1/20 0.37
ALOX15 P16050 1/20 0.37
TSHR P16473 1/20 0.37
MAPK1 P28482 1/20 0.37
HTT P42858 1/20 0.37
KMT2A Q03164 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Bicarbonate SCHEMBL1767911 0.99 HSP90AA1 (0.67) HSP90AA1HSP90AB1EGLN1KCNH2HRH4
Bicarbonate SCHEMBL1767988 0.97 HSP90AA1 (0.67) HSP90AA1HSP90AB1EGLN1KCNH2HRH4
Formic Acid SCHEMBL27886076 0.96 HSP90AA1 (0.64) HSP90AA1HSP90AB1EGLN1KCNH2HRH4
SCHEMBL1767936 0.96 HSP90AA1 (0.71) HSP90AA1HSP90AB1EGLN1KCNH2HRH4
Bicarbonate SCHEMBL1768011 0.94 HSP90AA1 (0.70) HSP90AA1HSP90AB1EGLN1KCNH2HRH4
Ethoxycarbonyl Group SCHEMBL28797508 0.89 HSP90AA1 (0.57) HSP90AA1HSP90AB1EGLN1NAMPT
SCHEMBL12273251 0.88 HSP90AA1 (0.64) HSP90AA1HSP90AB1EGLN1MEN1ALDH1A1
SCHEMBL16628709 0.83 HSP90AA1 (0.80) HSP90AA1HSP90AB1MEN1ALDH1A1LMNA
SCHEMBL16628686 0.82 HSP90AA1 (1.00) HSP90AA1HSP90AB1
SCHEMBL13180042 0.81 HSP90AA1 (0.73) HSP90AA1HSP90AB1MEN1ALDH1A1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2504314-A1 QUINAZOLINE DERIVATIVES Merck Patent GmbH (DE) 2012-10-03 EP disclosed
WO-2011060873-A1 QUINAZOLINE DERIVATIVES MERCK PATENT GMBH (DE) 2011-05-26 WO disclosed