SCHEMBL1768441

SCHEMBL1768441

NCc1noc(-c2c3c(Br)cccc3nn2CCn2ccnc2)n1

nearest known ligand 0.45

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 4/20 0.45
CYP2D6 P10635 3/20 0.45
SCN8A Q9UQD0 4/20 0.44
SCN1A P35498 2/20 0.44
SCN4A P35499 2/20 0.44
SCN5A Q14524 2/20 0.44
SCN9A Q15858 2/20 0.44
SCN2A Q99250 2/20 0.44
SCN3A Q9NY46 2/20 0.44
SCN10A Q9Y5Y9 2/20 0.44
CYP19A1 P11511 2/20 0.34
TBXAS1 P24557 1/20 0.34
CYP3A4 P08684 1/20 0.33
NOS1 P29475 1/20 0.32
HMOX2 P30519 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11896968 0.83 CYP1A2 (0.65) CYP1A2CYP2D6SCN8ASCN1ASCN4A
Ammonia Solution, Strong SCHEMBL1768336 0.82 CYP1A2 (0.64) CYP1A2CYP2D6SCN8ASCN1ASCN4A
SCHEMBL1768407 0.81 SCN8A (0.43) CYP1A2CYP2D6SCN8ASCN1ASCN4A
SCHEMBL1768561 0.81 CYP1A2 (0.49) CYP1A2CYP2D6SCN8ASCN1ASCN4A
SCHEMBL1768557 0.77 CYP1A2 (0.49) CYP1A2CYP2D6SCN8ASCN1ASCN4A
SCHEMBL1768299 0.73 SCN8A (0.69) CYP1A2CYP2D6SCN8ASCN1ASCN4A
SCHEMBL1768337 0.69 SCN8A (0.49) CYP1A2CYP2D6SCN8ASCN1ASCN4A
SCHEMBL11896994 0.69 SCN8A (0.67) CYP1A2CYP2D6SCN8ASCN1ASCN4A
SCHEMBL1768491 0.67 SCN8A (0.57) CYP1A2CYP2D6SCN8ASCN1ASCN4A
SCHEMBL12648966 0.67 SCN8A (0.76) CYP1A2CYP2D6SCN8ASCN1ASCN4A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2483270-A1 INDAZOLE DERIVATIVES AND THEIR USE FOR BLOCKADING VOLTAGE DEPENDENT SODIUM CHANNELS University College London (GB) 2012-08-08 EP disclosed
WO-2011061469-A1 INDAZOLE DERIVATIVES AND THEIR USE FOR BLOCKADING VOLTAGE DEPENDENT SODIUM CHANNELS UNIVERSITY COLLEGE LONDON (GB) 2011-05-26 WO disclosed