SCHEMBL1768461

SCHEMBL1768461

c1ccc(-c2cccc(P(c3ccccc3)c3ccccc3)c2P(c2ccccc2)c2ccccc2)cc1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TDP1 Q9NUW8 2/20 0.42
CYP3A4 P08684 1/20 0.42
CYP2A6 P11509 1/20 0.40
DRD1 P21728 2/20 0.39
ALDH1A1 P00352 4/20 0.35
HSD17B10 Q99714 2/20 0.35
HPGD P15428 1/20 0.35
BCL2L1 Q07817 1/20 0.35
MAPK1 P28482 1/20 0.35
ESR1 P03372 2/20 0.34
ESR2 Q92731 2/20 0.34
PTGS2 P35354 1/20 0.33
HTR6 P50406 1/20 0.33
PDCD1 Q15116 1/20 0.32
CD274 Q9NZQ7 1/20 0.32
HNF4A P41235 1/20 0.32
DPP4 P27487 1/20 0.32
BACE1 P56817 1/20 0.32
KDM4E B2RXH2 1/20 0.31
GAA P10253 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21333875 0.87 TDP1 (0.50) TDP1CYP3A4CYP2A6ALDH1A1HSD17B10
SCHEMBL29635182 0.83 TDP1 (0.50) TDP1CYP3A4CYP2A6DRD1ALDH1A1
SCHEMBL4004840 0.83 TDP1 (0.50) TDP1CYP3A4CYP2A6DRD1ALDH1A1
SCHEMBL28765143 0.83 CYP3A4 (0.55) TDP1CYP3A4DRD1ESR1ESR2
SCHEMBL7799500 0.81 TDP1 (0.48) TDP1CYP3A4CYP2A6DRD1ALDH1A1
SCHEMBL32685426 0.81 TDP1 (0.48) TDP1CYP3A4CYP2A6DRD1ALDH1A1
SCHEMBL28152682 0.80 TDP1 (0.42) TDP1CYP3A4CYP2A6DRD1ALDH1A1
SCHEMBL19664922 0.80 TDP1 (0.42) TDP1CYP3A4CYP2A6DRD1ALDH1A1
Bromide SCHEMBL6675138 0.79 TDP1 (0.46) TDP1CYP3A4CYP2A6DRD1ALDH1A1
SCHEMBL28427105 0.79 TDP1 (0.46) TDP1CYP3A4CYP2A6DRD1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 62 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112642489-B Homogeneous bimetallic complex catalyst, preparation method thereof and application thereof in preparation of aldehyde from alcohol 山东新和成药业有限公司 2022-09-20 CN claimed
CN-114181250-A Alkenyl phosphine compound and preparation method thereof 中国石油化工股份有限公司 2022-03-15 CN claimed
CN-107175134-B It is a kind of to be used to prepare 3-aminophenylacetylene or the composition of its salt and application thereof 成都西岭源药业有限公司 2018-03-23 CN claimed
EP-1341798-A1 CHIRAL DIPHOSPHINES AND THEIR METAL COMPLEXES PPG-Sipsy (FR) 2003-09-10 EP claimed
WO-2002040492-A1 CHIRAL DIPHOSPHINES AND THEIR METAL COMPLEXES PPG-SIPSY (FR) 2002-05-23 WO claimed
US-11739103-B2 Processes for preparing a pan-JAK inhibitor and related intermediate compounds Theravance Biopharma R&D LP, LLC (US) 2023-08-29 US disclosed
CN-114085200-B Method for preparing 2, 5-furandicarboxylic acid by using 2-furancarboxylic acid as raw material through one-pot method 华东师范大学 2023-03-14 CN disclosed
US-20220112219-A1 PROCESSES FOR PREPARING A PAN-JAK INHIBITOR AND RELATED INTERMEDIATE COMPOUNDS THERAVANCE BIOPHARMA R&D IP, LLC 2022-04-14 US disclosed
CN-114181250-A Alkenyl phosphine compound and preparation method thereof 中国石油化工股份有限公司 2022-03-15 CN disclosed
CN-114031494-A Method for preparing carboxylic acid by catalyzing reaction of unsaturated hydrocarbon and formic acid by using catalyst containing noble metal compound 华东师范大学 2022-02-11 CN disclosed
CN-110105308-A Preparation method of vortioxetine 山东京卫制药有限公司 2019-08-09 CN disclosed
CN-110105309-A A kind of preparation method lying prostrate sulphur Xi Ting 山东京卫制药有限公司 2019-08-09 CN disclosed
WO-2013035650-A1 METHOD FOR PRODUCING ALPHA - HYDROXY KETONE COMPOUND SUMITOMO CHEMICAL COMPANY, LIMITED (JP) 2013-03-14 WO disclosed
EP-2379575-A1 HYDROPHOSPHORYLATION OF PHOSPHONOUS ACID DERIVATIVES FOR FLAME RETARDANTS Clariant International Ltd. (CH) 2011-10-26 EP disclosed
WO-2011061439-A1 CATALYTIC PHOSPHINATION METHOD UNIVERSITE DE STRASBOURG (FR) 2011-05-26 WO disclosed
WO-2010069421-A1 HYDROPHOSPHORYLATION OF PHOSPHONOUS ACID DERIVATIVES FOR FLAME RETARDANTS CLARIANT INTERNATIONAL LTD (CH) 2010-06-24 WO disclosed
WO-2006100606-A2 PREPARATION OF BETA-AMINO ACID PRECURSORS VIA INDIUM (III) MEDIATED MARKOVNIKOV ADDITION AND KNOEVENAGEL CONDENSATION WARNER-LAMBERT COMPANY LLC (US) 2006-09-28 WO disclosed
WO-2004084834-A2 CHIRAL POROUS METAL PHOSPHONATES FOR HETEROGENEOUS ASYMMETRIC CATALYSIS THE UNIVERSITY OF NORTH CAROLINA AT CHAPEL HILL (US) 2004-10-07 WO disclosed
EP-0975574-A1 PROCESS TO PREPARE A PENTENOIC ACID DERIVATIVE DSM N.V. (NL) 2000-02-02 EP disclosed
WO-1998038151-A1 PROCESS TO PREPARE A PENTENOIC ACID DERIVATIVE DSM N.V. (NL) 1998-09-03 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20220112219-A1 PROCESSES FOR PREPARING A PAN-JAK INHIBITOR AND RELATED INTERMEDIATE COMPOUNDS JAK1, JAK3, JAK2 TDP1 2495/4885CYP3A4 825/4885CYP2A6 2400/4885
US-11739103-B2 Processes for preparing a pan-JAK inhibitor and related intermediate compounds JAK1, JAK3, JAK2 TDP1 2495/4885CYP3A4 825/4885CYP2A6 2400/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.