SCHEMBL17685207

SCHEMBL17685207

COCN(c1cccc(-c2nc(N)sc2Br)c1F)S(=O)(=O)c1cc(F)ccc1F

nearest known ligand 0.34

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
BRAF P15056 10/20 0.34
MPL P40238 2/20 0.31
NR1I2 O75469 4/20 0.31
FBP1 P09467 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17296630 0.86 BRAF (0.37) BRAFNR1I2FBP1
SCHEMBL17684952 0.84 BRAF (0.31) BRAF
SCHEMBL17684953 0.84 BRAF (0.31) BRAF
SCHEMBL17296632 0.82 BRAF (0.35) BRAFNR1I2
SCHEMBL574938 0.79 NPC1 (0.36)
SCHEMBL574448 0.79 KDM4E (0.36)
SCHEMBL15198328 0.78 BRAF (0.32) BRAF
SCHEMBL574870 0.77 MEN1 (0.32)
SCHEMBL575025 0.77 AKT1 (0.32)
SCHEMBL15191973 0.76 BRAF (0.42) BRAFNR1I2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2678336-B1 THIAZOLYLPHENYL-BENZENESULFONAMIDO DERIVATIVES AS KINASE INHIBITORS NERVIANO MEDICAL SCIENCES SRL (IT) 2016-04-20 EP disclosed