SCHEMBL17689241

SCHEMBL17689241

[2H]C([2H])(C#C)N(C)C[C@H](Cl)Cc1ccccc1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAOB P27338 10/20 0.45
MAOA P21397 7/20 0.45
CYP1A2 P05177 3/20 0.45
TSHR P16473 3/20 0.45
CYP2D6 P10635 2/20 0.45
ADRA2B P18089 2/20 0.45
ADRA2C P18825 2/20 0.45
ADRA1A P35348 2/20 0.45
OPRK1 P41145 2/20 0.45
ADRA2A P08913 1/20 0.45
SNCA P37840 1/20 0.45
PKM P14618 1/20 0.45
MAPK1 P28482 1/20 0.44
KDM4E B2RXH2 1/20 0.44
PYCR1 P32322 3/20 0.42
LMNA P02545 2/20 0.42
CYP3A4 P08684 2/20 0.42
USP2 O75604 1/20 0.42
ALDH1A1 P00352 1/20 0.41
BLM P54132 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17689239 1.00 MAOB (0.45) MAOBMAOACYP1A2TSHRCYP2D6
SCHEMBL694708 0.84 MAOB (0.57) MAOBMAOACYP1A2TSHRCYP2D6
SCHEMBL2479514 0.84 MAOB (0.57) MAOBMAOACYP1A2TSHRCYP2D6
SCHEMBL694707 0.84 MAOB (0.57) MAOBMAOACYP1A2TSHRCYP2D6
SCHEMBL17689247 0.82 MAOB (0.46) MAOBMAOACYP1A2TSHRCYP2D6
SCHEMBL18756808 0.77 MC4R (0.42) MAOBMAOATSHRADRA2BADRA2C
Selegiline SCHEMBL15867127 0.73 MAOB (0.71) MAOBMAOACYP1A2TSHRCYP2D6
Selegiline SCHEMBL7728634 0.73 MAOB (0.71) MAOBMAOACYP1A2TSHRCYP2D6
Selegiline SCHEMBL7731437 0.72 MAOB (0.55) MAOBMAOACYP1A2TSHRCYP2D6
SCHEMBL20018127 0.72 MAOB (0.41) MAOBMAOACYP1A2TSHRCYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9314540-B2 Compounds for use in imaging, diagnosing and/or treatment of diseases of the central nervous system PIRAMAL IMAGING SA (CH) 2016-04-19 US disclosed