SCHEMBL17689686

SCHEMBL17689686

CCCCC(=CC1=C(C)C(=O)C(OC)=C(OC)C1=O)C(=O)NOC

nearest known ligand 0.90

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
APEX1 P27695 10/20 0.90
MAPT P10636 2/20 0.40
TDP1 Q9NUW8 2/20 0.40
ALDH1A1 P00352 1/20 0.40
THRB P10828 1/20 0.40
LMNA P02545 2/20 0.34
PGR P06401 1/20 0.34
CYP3A4 P08684 1/20 0.34
CYP2D6 P10635 1/20 0.34
CYP2C9 P11712 1/20 0.34
MAOA P21397 1/20 0.34
TBXA2R P21731 1/20 0.34
MAPK1 P28482 1/20 0.34
AVPR2 P30518 1/20 0.34
CYP2C19 P33261 1/20 0.34
HTR2B P41595 1/20 0.34
HTT P42858 1/20 0.34
PDE3A Q14432 1/20 0.34
SIRT2 Q8IXJ6 1/20 0.34
SLC29A1 Q99808 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17277628 0.95 APEX1 (1.00) APEX1MAPTTDP1ALDH1A1THRB
SCHEMBL15711340 0.95 APEX1 (1.00) APEX1MAPTTDP1ALDH1A1THRB
SCHEMBL17835134 0.85 APEX1 (0.67) APEX1
SCHEMBL14135227 0.85 APEX1 (0.67) APEX1
SCHEMBL3755865 0.85 APEX1 (1.00) APEX1MAPTTDP1ALDH1A1THRB
SCHEMBL3755868 0.85 APEX1 (1.00) APEX1MAPTTDP1ALDH1A1THRB
SCHEMBL13049451 0.81 APEX1 (1.00) APEX1MAPTTDP1ALDH1A1THRB
Apx-3330 SCHEMBL3758716 0.80 APEX1 (1.00) APEX1MAPTTDP1ALDH1A1THRB
Apx-3330 SCHEMBL3758719 0.80 APEX1 (1.00) APEX1MAPTTDP1ALDH1A1THRB
SCHEMBL15705626 0.80 APEX1 (0.70) APEX1MAPTTDP1ALDH1A1THRB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9315481-B2 Compounds and methods for treating leukemia INDIANA UNIVERSITY RESEARCH AND TECHNOLOGY CORPORATION (US) 2016-04-19 US disclosed