SCHEMBL1769873

SCHEMBL1769873

NC(=O)c1ccc2cc(Br)ccc2c1.O=C(O)c1ccc2cc(Br)ccc2c1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LCK P06239 1/20 0.55
PARP1 P09874 1/20 0.52
DHODH Q02127 1/20 0.49
PLAU P00749 3/20 0.49
SRD5A1 P18405 1/20 0.47
SRD5A2 P31213 1/20 0.47
KDM4E B2RXH2 3/20 0.47
PARP15 Q460N3 2/20 0.46
PARP10 Q53GL7 2/20 0.46
PIM1 P11309 1/20 0.45
LMNA P02545 1/20 0.43
SMN1; SMN2 Q16637 1/20 0.43
MEN1 O00255 1/20 0.42
ALDH1A1 P00352 1/20 0.42
MAPT P10636 1/20 0.42
KMT2A Q03164 1/20 0.42
GLA P06280 1/20 0.42
PARP14 Q460N5 1/20 0.41
CYP2A6 P11509 1/20 0.41
DGAT1 O75907 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL613558 0.93 LCK (0.62) LCKPARP1DHODHPLAUKDM4E
SCHEMBL203205 0.91 DHODH (0.55) DHODHSRD5A1SRD5A2KDM4EPIM1
SCHEMBL30020656 0.91 DHODH (0.55) DHODHSRD5A1SRD5A2KDM4EPIM1
Hydrochloric Acid SCHEMBL1001004 0.89 DHODH (0.54) DHODHSRD5A1SRD5A2KDM4EPIM1
SCHEMBL29771387 0.89 LCK (0.67) LCKPARP1DHODHPLAUKDM4E
SCHEMBL1163640 0.89 LCK (0.67) LCKPARP1DHODHPLAUKDM4E
SCHEMBL15774265 0.87 LCK (0.60) LCKPARP1DHODHPLAUKDM4E
SCHEMBL2049058 0.85 SRD5A1 (0.53) DHODHSRD5A1SRD5A2KDM4EPIM1
Methoxymethane SCHEMBL27807143 0.84 KDM4E (0.62) DHODHPLAUSRD5A1SRD5A2KDM4E
SCHEMBL10081752 0.81 PTPN1 (0.53) DHODHSRD5A1SRD5A2KDM4EPIM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011061168-A1 ARYL-PYRIDINE DERIVATIVES AS ALDOSTERONE SYNTHASE INHIBITORS NOVARTIS AG (CH) 2011-05-26 WO disclosed