SCHEMBL17707491

SCHEMBL17707491

CCCC1(C(=O)c2ccc3ccccc3n2)CCN(C(=O)O)CC1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2D6 P10635 1/20 0.50
SLC6A2 P23975 1/20 0.50
SLC6A4 P31645 1/20 0.50
SLC6A3 Q01959 1/20 0.50
TSHR P16473 1/20 0.44
GRIN2B Q13224 2/20 0.44
MGAM O43451 1/20 0.43
GAA P10253 3/20 0.42
ALDH1A1 P00352 3/20 0.41
MAPT P10636 2/20 0.41
CNR2 P34972 3/20 0.41
RAB9A P51151 2/20 0.40
SMN1; SMN2 Q16637 2/20 0.40
SCN5A Q14524 1/20 0.40
SCN9A Q15858 1/20 0.40
MAPK1 P28482 1/20 0.40
KDM4C Q9H3R0 1/20 0.40
MEN1 O00255 1/20 0.39
KMT2A Q03164 1/20 0.39
L3MBTL1 Q9Y468 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL413992 0.85 CYP2D6 (0.50) CYP2D6SLC6A2SLC6A4SLC6A3GAA
SCHEMBL413990 0.82 CYP2D6 (0.68) CYP2D6SLC6A2SLC6A4SLC6A3MGAM
SCHEMBL31388159 0.81 CYP2D6 (0.48) CYP2D6SLC6A2SLC6A4SLC6A3GAA
Hydrochloric Acid SCHEMBL445019 0.81 CYP2D6 (0.67) CYP2D6SLC6A2SLC6A4SLC6A3MGAM
SCHEMBL12585782 0.67 CYP2D6 (0.82) CYP2D6SLC6A2SLC6A4SLC6A3MGAM
SCHEMBL415120 0.67 CYP2D6 (1.00) CYP2D6SLC6A2SLC6A4SLC6A3MGAM
Quinaldic Acid SCHEMBL17255915 0.66 MGAM (0.82) MGAMGAAALDH1A1MAPTCNR2
SCHEMBL28665600 0.65 MGAM (0.58) MGAMGAAALDH1A1MAPTCNR2
SCHEMBL5239212 0.65 KDM4E (0.68) SLC6A4TSHRALDH1A1RAB9ASMN1; SMN2
SCHEMBL29931500 0.65 KDM4E (0.68) SLC6A4TSHRALDH1A1RAB9ASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2684871-B1 Heteroaryl pyrrolidinyl and piperidinyl ketone derivatives HOFFMANN LA ROCHE (CH) 2016-05-04 EP disclosed