SCHEMBL17707494

SCHEMBL17707494

CCCC1(C(=O)c2cc(Cl)c(C)s2)CCN(C(=O)O)C1

nearest known ligand 0.37

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CYP2D6 P10635 4/20 0.37
SLC6A2 P23975 4/20 0.37
SLC6A4 P31645 4/20 0.37
SLC6A3 Q01959 4/20 0.37
P4HB P07237 1/20 0.33
ALDH1A1 P00352 2/20 0.32
LMNA P02545 1/20 0.32
MAPK1 P28482 1/20 0.32
KCNH2 Q12809 1/20 0.32
MEN1 O00255 2/20 0.31
KMT2A Q03164 2/20 0.31
RAB9A P51151 1/20 0.30
SPR P35270 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL415621 0.85 CYP2D6 (0.38) CYP2D6SLC6A2SLC6A4SLC6A3MEN1
SCHEMBL415219 0.76 SLC6A2 (0.63) CYP2D6SLC6A2SLC6A4SLC6A3KCNH2
Hydrochloric Acid SCHEMBL444317 0.75 SLC6A2 (0.61) CYP2D6SLC6A2SLC6A4SLC6A3KCNH2
SCHEMBL413350 0.75 CYP2D6 (0.47) CYP2D6SLC6A2SLC6A4SLC6A3MEN1
SCHEMBL16453921 0.72 CYP4F2 (0.34) MEN1KMT2A
SCHEMBL16453920 0.69 CYP4F2 (0.39) P4HBALDH1A1LMNAMEN1KMT2A
SCHEMBL17707487 0.67 CYP2D6 (0.31) CYP2D6SLC6A2SLC6A4SLC6A3SPR
SCHEMBL414185 0.67 SLC6A2 (0.67) CYP2D6SLC6A2SLC6A4SLC6A3KCNH2
SCHEMBL18597661 0.67 SLC6A2 (0.51) CYP2D6SLC6A2SLC6A4SLC6A3P4HB
SCHEMBL31388169 0.66 ACKR3 (0.52) CYP2D6SLC6A2SLC6A4SLC6A3RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2684871-B1 Heteroaryl pyrrolidinyl and piperidinyl ketone derivatives HOFFMANN LA ROCHE (CH) 2016-05-04 EP disclosed