SCHEMBL17786331

SCHEMBL17786331

COc1cc(O)c(C(C)=O)cc1N

nearest known ligand 0.72

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
HTT P42858 2/20 0.72
CYP3A4 P08684 5/20 0.49
ALDH1A1 P00352 3/20 0.49
MAPK1 P28482 2/20 0.49
HPGD P15428 2/20 0.49
HMGCR P04035 1/20 0.47
LMNA P02545 3/20 0.44
KDM4E B2RXH2 2/20 0.44
L3MBTL1 Q9Y468 2/20 0.44
PKM P14618 1/20 0.44
EP300 Q09472 1/20 0.43
USP2 O75604 1/20 0.43
SMN1; SMN2 Q16637 1/20 0.43
MAPT P10636 2/20 0.42
RECQL P46063 1/20 0.42
HSD17B10 Q99714 1/20 0.42
POLB P06746 1/20 0.42
GAA P10253 4/20 0.41
S100B P04271 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17774729 0.85 HTT (0.52) HTTCYP3A4ALDH1A1HPGDHMGCR
SCHEMBL6371675 0.85 CYP3A4 (0.55) HTTCYP3A4ALDH1A1LMNAKDM4E
SCHEMBL3661837 0.84 HTT (1.00) HTTCYP3A4ALDH1A1MAPK1HPGD
SCHEMBL30398255 0.84 HTT (1.00) HTTCYP3A4ALDH1A1MAPK1HPGD
SCHEMBL31175997 0.82 HTT (0.81) HTTCYP3A4ALDH1A1MAPK1HPGD
SCHEMBL14780513 0.82 HTT (0.81) HTTCYP3A4ALDH1A1MAPK1HPGD
SCHEMBL26027709 0.81 KDM4E (0.56) HTTCYP3A4ALDH1A1LMNAKDM4E
SCHEMBL22222472 0.80 HTT (0.46) HTTCYP3A4ALDH1A1MAPK1LMNA
SCHEMBL5526244 0.80 HTT (0.52) HTTCYP3A4ALDH1A1MAPK1HPGD
SCHEMBL1545430 0.79 HTT (0.81) HTTCYP3A4ALDH1A1MAPK1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2016083490-A1 COMPOUNDS FOR THE TREATMENT OF AMYLOID-ASSOCIATED DISEASES REMYND NV (BE) 2016-06-02 WO disclosed