SCHEMBL17801093

SCHEMBL17801093

CS(=O)(=O)Nc1cccc(-c2n[nH]c3ccc(-c4n[nH]c(C5CCCN5C(=O)O)n4)cc23)c1

nearest known ligand 0.63

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
CPT1A P50416 16/20 0.63
CPT2 P23786 11/20 0.63
CSNK1D P48730 1/20 0.49
CPT1B Q92523 1/20 0.47
AAK1 Q2M2I8 1/20 0.45
HCRTR1 O43613 2/20 0.44
HCRTR2 O43614 2/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17801091 0.84 CPT1A (0.60) CPT1ACPT2CPT1BHCRTR1HCRTR2
SCHEMBL17801081 0.84 CPT1A (0.46) CPT1ACPT2CPT1BHCRTR1HCRTR2
SCHEMBL17801057 0.81 CPT1A (0.51) CPT1ACPT2CPT1BHCRTR1HCRTR2
SCHEMBL17801049 0.79 CPT1A (0.52) CPT1ACPT2CPT1BHCRTR1HCRTR2
SCHEMBL17801046 0.79 CPT1A (0.45) CPT1ACPT2CPT1BHCRTR1HCRTR2
SCHEMBL3551630 0.77 CPT1A (1.00) CPT1ACPT2CPT1B
SCHEMBL3551631 0.77 CPT1A (1.00) CPT1ACPT2CPT1B
SCHEMBL17801010 0.75 HCRTR2 (0.44) CPT1ACPT2CPT1BHCRTR1HCRTR2
SCHEMBL17801054 0.75 CPT1A (0.55) CPT1ACPT2CPT1BHCRTR1HCRTR2
SCHEMBL5377458 0.71 CSNK1D (0.55) CSNK1DAAK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2016089977-A1 SUBSTITUTED INDAZOLE COMPOUNDS, COMPOSITIONS THEREOF, AND METHODS OF TREATMENT THEREWITH CELGENE CORPORATION (US) 2016-06-09 WO disclosed