SCHEMBL17806502

SCHEMBL17806502

Cn1cnc2c(F)c(Nc3ccc(Br)cc3F)c(C(=O)NOCCOS(N)(=O)=O)cc21

nearest known ligand 0.80

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
MAP2K1 Q02750 20/20 0.80
MAP2K2 P36507 2/20 0.80
ABCB11 O95342 1/20 0.80
NQO2 P16083 1/20 0.80
SMC2 O95347 1/20 0.68
EGFR P00533 1/20 0.68
CSNK2A2 P19784 1/20 0.68
SMC1A Q14683 1/20 0.68
AAK1 Q2M2I8 1/20 0.68
Q6ZSR9 Q6ZSR9 1/20 0.68
BMP2K Q9NSY1 1/20 0.68
BRAF P15056 5/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17806506 0.92 MAP2K1 (0.81) MAP2K1MAP2K2ABCB11NQO2SMC2
SCHEMBL29990127 0.90 MAP2K1 (0.88) MAP2K1MAP2K2ABCB11NQO2SMC2
SCHEMBL25189605 0.90 MAP2K1 (0.88) MAP2K1MAP2K2ABCB11NQO2SMC2
SCHEMBL25480020 0.89 MAP2K1 (0.84) MAP2K1MAP2K2ABCB11NQO2SMC2
SCHEMBL15704258 0.89 MAP2K1 (0.84) MAP2K1MAP2K2ABCB11NQO2SMC2
Binimetinib SCHEMBL570088 0.89 MAP2K1 (1.00) MAP2K1MAP2K2ABCB11NQO2SMC2
Binimetinib SCHEMBL29363187 0.89 MAP2K1 (1.00) MAP2K1MAP2K2ABCB11NQO2SMC2
SCHEMBL29199685 0.89 MAP2K1 (0.83) MAP2K1MAP2K2ABCB11NQO2SMC2
SCHEMBL15647087 0.88 MAP2K1 (0.81) MAP2K1MAP2K2ABCB11NQO2SMC2
SCHEMBL29992273 0.88 MAP2K1 (0.81) MAP2K1MAP2K2ABCB11NQO2SMC2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2016089208-A2 SULFONAMIDE, SULFAMATE AND SULFAMIDE DERIVATIVES OF ANTI-CANCER AGENTS STICHTING MAASTRICHT RADIATION ONCOLOGY "MAASTRO-CLINIC" (NL) 2016-06-09 WO disclosed