SCHEMBL17812934

SCHEMBL17812934

CC[C@@H]1CC[C@@H](O)CN1C(=O)c1ccccc1-n1nccn1

nearest known ligand 0.61

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
HCRTR2 O43614 20/20 0.61
HCRTR1 O43613 18/20 0.61
CYP3A4 P08684 6/20 0.56

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17803665 0.89 HCRTR1 (0.61) HCRTR2HCRTR1CYP3A4
SCHEMBL17812932 0.89 HCRTR1 (0.61) HCRTR2HCRTR1CYP3A4
SCHEMBL7918180 0.84 HCRTR2 (0.65) HCRTR2HCRTR1
SCHEMBL7915973 0.84 HCRTR2 (0.65) HCRTR2HCRTR1
SCHEMBL2291824 0.84 HCRTR2 (0.65) HCRTR2HCRTR1
SCHEMBL17812933 0.82 HCRTR2 (0.51) HCRTR2HCRTR1CYP3A4
SCHEMBL17812927 0.82 HCRTR2 (0.51) HCRTR2HCRTR1CYP3A4
SCHEMBL17803651 0.81 HCRTR2 (0.48) HCRTR2HCRTR1
SCHEMBL19564500 0.81 HCRTR2 (0.51) HCRTR2HCRTR1CYP3A4
SCHEMBL17812946 0.81 HCRTR2 (0.59) HCRTR2HCRTR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2016086358-A1 HYDROXYMETHYL PIPERIDINE OREXIN RECEPTOR ANTAGONISTS MERCK SHARP & DOHME CORP. (US) 2016-06-09 WO disclosed