SCHEMBL17813396

SCHEMBL17813396

O=C(Nc1ccc2c(c1)CCCN(C1CC1)C2)OCc1ccccc1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PSEN1 P49768 1/20 0.49
PSEN2 P49810 1/20 0.49
APH1B Q8WW43 1/20 0.49
NCSTN Q92542 1/20 0.49
APH1A Q96BI3 1/20 0.49
PSENEN Q9NZ42 1/20 0.49
HRH3 Q9Y5N1 4/20 0.48
TMEM97 Q5BJF2 5/20 0.48
SIGMAR1 Q99720 5/20 0.48
NPC1 O15118 2/20 0.47
RAB9A P51151 2/20 0.47
ALDH1A1 P00352 1/20 0.47
TP53 P04637 1/20 0.47
MAPT P10636 1/20 0.47
TSHR P16473 1/20 0.47
ATM Q13315 1/20 0.47
SMN1; SMN2 Q16637 1/20 0.47
MGLL Q99685 1/20 0.46
HTR1A P08908 2/20 0.46
HRH2 P25021 2/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17797537 0.96 TMEM97 (0.52) PSEN1PSEN2APH1BNCSTNAPH1A
SCHEMBL14429561 0.85 HRH3 (0.59) PSEN1PSEN2APH1BNCSTNAPH1A
SCHEMBL30981352 0.85 NPC1 (0.47) PSEN1PSEN2APH1BNCSTNAPH1A
SCHEMBL17797663 0.83 TMEM97 (0.55) PSEN1PSEN2APH1BNCSTNAPH1A
SCHEMBL9447608 0.82 NPC1 (0.65) PSEN1PSEN2APH1BNCSTNAPH1A
SCHEMBL17797709 0.81 KMT2A (0.46) NPC1RAB9AALDH1A1TP53MAPT
SCHEMBL17797565 0.80 TMEM97 (0.54) PSEN1PSEN2APH1BNCSTNAPH1A
SCHEMBL6296040 0.80 TMPRSS2 (0.56) PSEN1PSEN2APH1BNCSTNAPH1A
SCHEMBL30981397 0.80 TMEM97 (0.43) PSEN1PSEN2APH1BNCSTNAPH1A
SCHEMBL6292442 0.79 TMEM97 (0.62) HRH3TMEM97SIGMAR1NPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2016090079-A1 HETEROARYL COMPOUNDS AND USES THEREOF CELGENE AVILOMICS RESEARCH, INC. (US) 2016-06-09 WO disclosed