SCHEMBL17822136

SCHEMBL17822136

c1cc(Nc2ncc3nc[nH]c3n2)n[nH]1

nearest known ligand 0.34

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
CDK1 P06493 6/20 0.34
CDK2 P24941 1/20 0.33
TNIK Q9UKE5 1/20 0.31
ULK1 O75385 1/20 0.31
ULK2 Q8IYT8 1/20 0.31
KDM4E B2RXH2 1/20 0.30
ALDH1A1 P00352 1/20 0.30
GLA P06280 1/20 0.30
GAA P10253 1/20 0.30
HPGD P15428 1/20 0.30
HSD17B10 Q99714 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17822137 0.78 CDK2 (0.58) CDK1CDK2TNIKKDM4EALDH1A1
SCHEMBL4551624 0.76 FLT3 (0.44) CDK1CDK2ALDH1A1HPGD
SCHEMBL165738 0.74 ROCK1 (0.45) CDK1CDK2KDM4E
SCHEMBL3026520 0.73 CDK2 (0.60) CDK1CDK2
SCHEMBL4480587 0.70 KDM4E (0.33) CDK1CDK2KDM4EALDH1A1GLA
SCHEMBL28506082 0.70
SCHEMBL5828206 0.70 KDM4E (0.36) CDK1CDK2KDM4EALDH1A1GLA
SCHEMBL30850504 0.70 EGFR (0.36) CDK1CDK2ULK1KDM4EALDH1A1
SCHEMBL30677393 0.70 KDM4E (0.36) CDK1CDK2KDM4EALDH1A1GLA
SCHEMBL5072697 0.70 EGFR (0.36) CDK1CDK2ULK1KDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2016091916-A1 PYRAZOLYLAMINOPURINES AS ITK INHIBITORS F. HOFFMANN-LA ROCHE AG (CH) 2016-06-16 WO disclosed
WO-2016091916-A1 PYRAZOLYLAMINOPURINES AS ITK INHIBITORS F. HOFFMANN-LA ROCHE AG (CH) 2016-06-16 WO disclosed