SCHEMBL17827945

SCHEMBL17827945

Cc1ccc2ncnc(N3CCCCC3c3cc4nc(N5CCCC5)ccn4n3)c2c1

nearest known ligand 0.57

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 2/20 0.39
RAB9A P51151 2/20 0.39
SMN1; SMN2 Q16637 2/20 0.39
KDM4E B2RXH2 1/20 0.39
TP53 P04637 1/20 0.39
GAA P10253 1/20 0.39
MAPT P10636 1/20 0.39
ALOX15 P16050 1/20 0.39
CASP1 P29466 1/20 0.39
HTT P42858 1/20 0.39
CASP7 P55210 1/20 0.39
HSD17B10 Q99714 1/20 0.39
ALDH1A1 P00352 1/20 0.39
NPSR1 Q6W5P4 1/20 0.39
CHRM4 P08173 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17827760 1.00 NPC1 (0.39) NPC1RAB9ASMN1; SMN2KDM4ETP53
SCHEMBL17823209 0.91 CHRM4 (0.37) CHRM4
SCHEMBL17823272 0.91 CHRM4 (0.37) CHRM4
SCHEMBL19677562 0.91 CHRM4 (0.37) CHRM4
SCHEMBL17823234 0.91 CHRM4 (0.37) CHRM4
SCHEMBL19677563 0.91 CHRM4 (0.37) CHRM4
SCHEMBL17823276 0.85 CHRM4 (0.40) CHRM4
SCHEMBL17823277 0.85
SCHEMBL19665196 0.84 MAP4K4 (0.33)
SCHEMBL19677558 0.83 MAP4K4 (0.47)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2016091774-A1 PIPERIDINE SUBSTITUTED PYRAZOLO[1,5-A]PYRIMIDINE DERIVATIVES WITH INHIBITORY ACTIVITY ON THE REPLICATION OF THE RESPIRATORY SYNCYTIAL VIRUS (RSV) JANSSEN SCIENCES IRELAND UC (IE) 2016-06-16 WO disclosed