SCHEMBL17844353

SCHEMBL17844353

O=S1(=O)CCCCN1c1ccccc1

nearest known ligand 0.64

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
POLB P06746 1/20 0.64
CA1 P00915 1/20 0.60
CA2 P00918 1/20 0.60
CA6 P23280 1/20 0.60
OPRK1 P41145 1/20 0.60
CA7 P43166 1/20 0.60
CA9 Q16790 1/20 0.60
MAPT P10636 1/20 0.55
TP53 P04637 1/20 0.47
AKR1C3 P42330 1/20 0.44
SLC9A3 P48764 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12209941 0.94 POLB (0.57) POLBCA1CA2CA6OPRK1
SCHEMBL31195399 0.81 CA1 (0.61) POLBCA1CA2CA6OPRK1
SCHEMBL8262169 0.81 CA1 (0.61) POLBCA1CA2CA6OPRK1
SCHEMBL1030597 0.81 CA1 (0.66) POLBCA1CA2CA6OPRK1
SCHEMBL8358594 0.81 CA1 (0.61) POLBCA1CA2CA6OPRK1
SCHEMBL25845301 0.81 CA1 (0.61) POLBCA1CA2CA6OPRK1
SCHEMBL5362725 0.80 POLB (0.68) POLBCA1CA2CA6OPRK1
Hydrochloric Acid SCHEMBL3544398 0.79 CA1 (0.64) POLBCA1CA2CA6OPRK1
SCHEMBL15683644 0.79 CA1 (0.59) POLBCA1CA2CA6OPRK1
SCHEMBL10053487 0.79 POLB (0.62) POLBCA1CA2CA6OPRK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3233849-A1 HETEROARYLALKYLENE ARYL SULTAM DERIVATIVES AS RORc MODULATORS F. Hoffmann-La Roche AG (CH) 2017-10-25 EP disclosed
WO-2016096936-A1 HETEROARYLALKYLENE ARYL SULTAM DERIVATIVES AS RORc MODULATORS F. HOFFMANN-LA ROCHE AG (CH) 2016-06-23 WO disclosed