SCHEMBL17845138

SCHEMBL17845138

O=Cc1c(-c2ccc(F)cc2)sc2cc(O)ccc12

nearest known ligand 0.58

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 17/20 0.58
APP P05067 1/20 0.44
SULT1A1 P50225 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16346118 0.92 ESR1 (0.52) ESR1
SCHEMBL30898315 0.92 ESR1 (0.52) ESR1
SCHEMBL18150143 0.92 ESR1 (0.67) ESR1
SCHEMBL18150144 0.88 ESR1 (0.49) ESR1APPSULT1A1
SCHEMBL28445468 0.79 APP (0.48) ESR1APP
SCHEMBL30610954 0.79 ESR1 (0.60) ESR1APPSULT1A1
SCHEMBL19143729 0.79 ESR1 (0.60) ESR1APPSULT1A1
SCHEMBL20425311 0.79 ESR1 (0.60) ESR1APPSULT1A1
SCHEMBL31683627 0.77 ESR1 (0.81) ESR1
SCHEMBL8631942 0.77 ESR1 (0.81) ESR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-107406424-B Estrogen receptor modulators and uses thereof 豪夫迈·罗氏有限公司 2020-08-25 CN disclosed
EP-3233828-A1 ESTROGEN RECEPTOR MODULATORS AND USES THEREOF F. Hoffmann-La Roche AG (CH) 2017-10-25 EP disclosed
WO-2016097071-A1 ESTROGEN RECEPTOR MODULATORS AND USES THEREOF F. HOFFMANN-LA ROCHE AG (CH) 2016-06-23 WO disclosed