SCHEMBL17845166

SCHEMBL17845166

O=Cc1cc(F)c(OCCN2CC(CF)C2)c(-c2c(-c3ccccc3Cl)noc2-c2ccc(OC3CCCCO3)cc2)c1

nearest known ligand 0.32

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 14/20 0.32
TNK2 Q07912 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17845085 0.86 ESR1 (0.38) ESR1TNK2
SCHEMBL17845119 0.80 ESR1 (0.38) ESR1
SCHEMBL21780917 0.74 ESR1 (0.48) ESR1
SCHEMBL17845111 0.72 ESR1 (0.37) ESR1
SCHEMBL17858145 0.72 ESR1 (0.48) ESR1
SCHEMBL17845094 0.70 PTGS1 (0.38) TNK2
SCHEMBL17845123 0.69 ESR1 (0.46) ESR1
SCHEMBL17845162 0.69 ESR1 (0.46) ESR1
SCHEMBL17845161 0.69 ESR1 (0.46) ESR1
SCHEMBL17845087 0.68 TNK2 (0.39) TNK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3233828-A1 ESTROGEN RECEPTOR MODULATORS AND USES THEREOF F. Hoffmann-La Roche AG (CH) 2017-10-25 EP disclosed
WO-2016097071-A1 ESTROGEN RECEPTOR MODULATORS AND USES THEREOF F. HOFFMANN-LA ROCHE AG (CH) 2016-06-23 WO disclosed