SCHEMBL17846803

SCHEMBL17846803

CCN(C(=O)c1c(F)cccc1-n1nccn1)C(C)N(C)c1cc(C#N)ccn1

nearest known ligand 0.70

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
HCRTR2 O43614 20/20 0.70
HCRTR1 O43613 19/20 0.70

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17846802 0.82 HCRTR1 (1.00) HCRTR2HCRTR1
SCHEMBL17846790 0.81 HCRTR1 (0.68) HCRTR2HCRTR1
SCHEMBL17846792 0.70 HCRTR1 (0.67) HCRTR2HCRTR1
SCHEMBL17846752 0.70 HCRTR1 (1.00) HCRTR2HCRTR1
SCHEMBL17846729 0.70 HCRTR1 (1.00) HCRTR2HCRTR1
SCHEMBL17846706 0.70 HCRTR2 (1.00) HCRTR2HCRTR1
SCHEMBL17846782 0.69 HCRTR1 (0.67) HCRTR2HCRTR1
SCHEMBL19689855 0.68 HCRTR1 (1.00) HCRTR2HCRTR1
SCHEMBL17846756 0.67 HCRTR1 (1.00) HCRTR2HCRTR1
SCHEMBL17846773 0.67 HCRTR2 (1.00) HCRTR2HCRTR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2016100161-A1 ETHYLDIAMINE OREXIN RECEPTOR ANTAGONISTS MERCK SHARP & DOHME CORP. (US) 2016-06-23 WO claimed