SCHEMBL17847972

SCHEMBL17847972

COc1ccc2c(c1)C(CC(=O)N(C)Cc1ccco1)=C(C)C2=Cc1cc(OC)c(O)c(OC)c1

nearest known ligand 0.42

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
PPARG P37231 2/20 0.42
TSHR P16473 6/20 0.41
LCK P06239 1/20 0.41
L3MBTL1 Q9Y468 2/20 0.41
ALDH1A1 P00352 5/20 0.39
KDM4E B2RXH2 5/20 0.39
MAPT P10636 3/20 0.39
APEX1 P27695 1/20 0.39
RXRA P19793 1/20 0.38
HPGD P15428 4/20 0.37
HSD17B10 Q99714 1/20 0.37
NPSR1 Q6W5P4 1/20 0.37
GAA P10253 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17847971 1.00 PPARG (0.42) PPARGTSHRLCKL3MBTL1ALDH1A1
SCHEMBL17847730 0.93 PPARG (0.42) PPARGTSHRL3MBTL1ALDH1A1KDM4E
SCHEMBL17847728 0.93 PPARG (0.42) PPARGTSHRL3MBTL1ALDH1A1KDM4E
SCHEMBL22215267 0.91 PPARG (0.40) PPARGTSHRL3MBTL1ALDH1A1KDM4E
SCHEMBL19857213 0.91 PPARG (0.47) PPARGTSHRALDH1A1KDM4EMAPT
SCHEMBL17853928 0.91 PPARG (0.47) PPARGTSHRALDH1A1KDM4EMAPT
SCHEMBL19017441 0.89 PPARG (0.42) PPARGTSHRLCKL3MBTL1ALDH1A1
SCHEMBL17847950 0.86 PPARG (0.46) PPARGTSHRLCKL3MBTL1ALDH1A1
SCHEMBL17847945 0.86 PPARG (0.46) PPARGTSHRLCKL3MBTL1ALDH1A1
SCHEMBL17854864 0.86 PPARG (0.46) PPARGTSHRLCKL3MBTL1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 10 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3666268-A1 METHOD OF TREATING OR PREVENTING RAS-MEDIATED DISEASES ADT Pharmaceuticals, LLC (US) 2020-06-17 EP claimed
US-11198679-B2 Method of treating or preventing Ras-mediated diseases ADT PHARMACEUTICALS, LLC (US) 2021-12-14 US disclosed
CN-107466232-B Methods of treating or preventing RAS-mediated diseases ADT制药有限责任公司 2021-06-29 CN disclosed
US-20200223817-A1 METHOD OF TREATING OR PREVENTING RAS-MEDIATED DISEASES ADT PHARMACEUTICALS, LLC (US) 2020-07-16 US disclosed
EP-3666268-A1 METHOD OF TREATING OR PREVENTING RAS-MEDIATED DISEASES ADT Pharmaceuticals, LLC (US) 2020-06-17 EP disclosed
EP-3233071-B1 METHOD OF TREATING OR PREVENTING RAS-MEDIATED DISEASES ADT PHARMACEUTICALS LLC (US) 2019-09-18 EP disclosed
US-20180251443-A9 METHOD OF TREATING OR PREVENTING RAS-MEDIATED DISEASES ADT PHARMACEUTICALS, LLC 2018-09-06 US disclosed
US-20180044314-A1 METHOD OF TREATING OR PREVENTING RAS-MEDIATED DISEASES ADT PHARMACEUTICALS INC (US) 2018-02-15 US disclosed
EP-3233071-A1 METHOD OF TREATING OR PREVENTING RAS-MEDIATED DISEASES ADT Pharmaceuticals, Inc. (US) 2017-10-25 EP disclosed
WO-2016100546-A1 METHOD OF TREATING OR PREVENTING RAS-MEDIATED DISEASES ADT PHARMACEUTICALS, INC. (US) 2016-06-23 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20180251443-A9 METHOD OF TREATING OR PREVENTING RAS-MEDIATED DISEASES KRAS, NRAS, HRAS PPARG 1654/4885TSHR 697/4885LCK 1962/4885
US-11198679-B2 Method of treating or preventing Ras-mediated diseases KRAS, NRAS, HRAS PPARG 1654/4885TSHR 697/4885LCK 1962/4885
US-20180044314-A1 METHOD OF TREATING OR PREVENTING RAS-MEDIATED DISEASES KRAS, NRAS, HRAS PPARG 1654/4885TSHR 697/4885LCK 1962/4885
US-20200223817-A1 METHOD OF TREATING OR PREVENTING RAS-MEDIATED DISEASES KRAS, NRAS, HRAS PPARG 1654/4885TSHR 697/4885LCK 1962/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.